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PRMT1 is a novel molecular therapeutic target for clear cell renal cell carcinoma 期刊论文
THERANOSTICS, 2021, 卷号: 11, 期号: 11, 页码: 5387-5403
作者:  Wang, Jianfeng;  Wang, Chen;  Xu, Pan;  Li, Xiao;  Lu, Yongning
收藏  |  浏览/下载:131/0  |  提交时间:2021/05/24
Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening 期刊论文
RSC ADVANCES, 2019, 卷号: 9, 期号: 9, 页码: 4917-4924
作者:  Tao, Hongru;  Wang, Jun;  Lu, Wenchao;  Zhang, Rukang;  Xie, Yiqian
收藏  |  浏览/下载:43/0  |  提交时间:2020/07/01
Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 8888-8905
作者:  Wang, Chen;  Jiang, Hao;  Jin, Jia;  Xie, Yiqian;  Chen, Zhifeng
收藏  |  浏览/下载:116/0  |  提交时间:2019/01/08
Machine-Learning-Assisted Approach for Discovering Novel Inhibitors Targeting Bromodomain-Containing Protein 4 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017, 卷号: 57, 期号: 7, 页码: 1677-1690
作者:  Xing, Jing;  Lu, Wenchao;  Liu, Rongfeng;  Wang, Yulan;  Xie, Yiqian
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay 期刊论文
MEDCHEMCOMM, 2017, 卷号: 8, 期号: 6, 页码: 1322-1331
作者:  Chen, Zhifeng;  Zhang, Hao;  Liu, Shien;  Xie, Yiqian;  Jiang, Hao
收藏  |  浏览/下载:91/0  |  提交时间:2019/01/08
Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 20, 页码: 8166-8181
作者:  Meng, Fanwang;  Cheng, Sufang;  Ding, Hong;  Liu, Shien;  Liu, Yan
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Discovery of two aminoglycoside antibiotics as inhibitors targeting the menin-mixed lineage leukaemia interface 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 9, 页码: 2090-2093
作者:  Li, Lianchun;  Zhou, Ran;  Geng, Heji;  Yue, Liyan;  Ye, Fei
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Virtual screening and biological evaluation of novel small molecular inhibitors against protein arginine methyltransferase 1 (PRMT1) 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2014, 卷号: 12, 期号: 47, 页码: 9665-9673
作者:  Xie, Yiqian;  Zhou, Ran;  Lian, Fulin;  Liu, Yan;  Chen, Limin
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Boc5, a Non-Peptidic Glucagon-Like Peptide-1 Receptor Agonist, Invokes Sustained Glycemic Control and Weight Loss in Diabetic Mice 期刊论文
PLOS ONE, 2008, 卷号: 3, 期号: 8
作者:  Su, Haoran;  He, Min;  Li, Hongmei;  Liu, Qing;  Wang, Jia
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08


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