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科研机构
北京大学 [51]
内容类型
期刊论文 [49]
其他 [2]
发表日期
2017 [5]
2016 [8]
2015 [1]
2014 [7]
2013 [5]
2012 [3]
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专题:北京大学
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NF-kappa B signaling and cell-fate decision induced by a fast-dissociating tumor necrosis factor mutant
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017
Zhang, Xiaoling
;
Yin, Ning
;
Guo, Annan
;
Zhang, Qi
;
Zhang, Yalei
;
Xu, Youjun
;
Liu, Hongbo
;
Tang, Bo
;
Lai, Luhua
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
NF-kappa B signaling dynamics
TNF
Receptor-ligand binding kinetics
Gene expression
Biased activation
Apoptosis
GENE-EXPRESSION
DYNAMICS
SPECIFICITY
DETERMINES
KINETICS
ALPHA
TNF
Tuning SpyTag-SpyCatcher mutant pairs toward orthogonal reactivity encryption
期刊论文
CHEMICAL SCIENCE, 2017
Liu, Yajie
;
Liu, Dong
;
Yang, Wei
;
Wu, Xia-Ling
;
Lai, Luhua
;
Zhang, Wen-Bin
收藏
  |  
浏览/下载:114/0
  |  
提交时间:2017/12/03
PROTEINS IN-VIVO
DIRECTED EVOLUTION
GIANT MOLECULES
CHEMISTRY
DESIGN
TOPOLOGY
ENZYME
BOND
PharmMapper 2017 update: a web server for potential drug target identification with a comprehensive target pharmacophore database
期刊论文
NUCLEIC ACIDS RESEARCH, 2017
Wang, Xia
;
Shen, Yihang
;
Wang, Shiwei
;
Li, Shiliang
;
Zhang, Weilin
;
Liu, Xiaofeng
;
Lai, Luhua
;
Pei, Jianfeng
;
Li, Honglin
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
DOCKING APPROACH
PROTEIN TARGETS
GENERATION
PREDICTION
MOLECULES
SEARCH
DESIGN
PHARMACOLOGY
POCKET
Origin of the Reflectin Gene and Hierarchical Assembly of Its Protein
期刊论文
CURRENT BIOLOGY, 2017
Guan, Zhe
;
Cai, Tiantian
;
Liu, Zhongmin
;
Dou, Yunfeng
;
Hu, Xuesong
;
Zhang, Peng
;
Sun, Xin
;
Li, Hongwei
;
Kuang, Yao
;
Zhai, Qiran
;
Ruan, Hao
;
Li, Xuanxuan
;
Li, Zeyang
;
Zhu, Qihui
;
Mai, Jingeng
;
Wang, Qining
;
Lai, Luhua
;
Ji, Jianguo
;
Liu, Haiguang
;
Xia, Bin
;
Jiang, Taijiao
;
Luo, Shu-Jin
;
Wang, Hong-Wei
;
Xie, Can
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
CEPHALOPOD DYNAMIC CAMOUFLAGE
NEIGHBOR-JOINING METHOD
STRUCTURAL COLORATION
LOLLIGUNCULA-BREVIS
SQUID
IRIDESCENCE
EVOLUTION
BIOPHOTONICS
PHYLOGENIES
SCATTERING
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
Structure-based Inhibitor Design for the Intrinsically Disordered Protein c-Myc
期刊论文
SCIENTIFIC REPORTS, 2016
Yu, Chen
;
Niu, Xiaogang
;
Jin, Fan
;
Liu, Zhirong
;
Jin, Changwen
;
Lai, Luhua
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
SMALL-MOLECULE INHIBITOR
MYC/MAX DIMERIZATION
DRUG DESIGN
UNSTRUCTURED PROTEINS
SELECTIVE-INHIBITION
ACCURATE DOCKING
NMR-SPECTROSCOPY
LEUCINE-ZIPPER
BINDING
MODEL
Novel Inhibitors of Toxin HipA Reduce Multidrug Tolerant Persisters
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2016
Li, Tongqing
;
Yin, Ning
;
Liu, Hongbo
;
Pei, Jianfeng
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
Persistence
toxin-antitoxin (TA) module
HipA (high persistence A)
drug discovery
ESCHERICHIA-COLI
BACTERIAL PERSISTENCE
MOLECULAR-MECHANISMS
CELLS
Discovery of Non-ATP-Competitive Inhibitors of Polo-like Kinase1
期刊论文
CHEMMEDCHEM, 2016
Yun, Taikangxiang
;
Qin, Tan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
inhibitors
kinase domain
non-ATP binding site
polo-like kinase1
virtual screening
1 PLK1 INHIBITORS
P38 MAP KINASE
CANCER-THERAPY
BINDING-SITE
BOX DOMAIN
PROTEIN
POLO-LIKE-KINASE-1
IDENTIFICATION
APOPTOSIS
DESIGN
Discovery of Novel 15-Lipoxygenase Activators To Shift the Human Arachidonic Acid Metabolic Network toward Inflammation Resolution
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Meng, Hu
;
McClendon, Christopher L.
;
Dai, Ziwei
;
Li, Kenan
;
Zhang, Xiaoling
;
He, Shan
;
Shang, Erchang
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
INHIBITION
ENZYMES
MODEL
SITE
BIOSYNTHESIS
PROSTACYCLIN
PROTEINS
EFFECTOR
SYNTHASE
LIGANDS
De novo design of helical peptides to inhibit tumor necrosis factor-alpha by disrupting its trimer formation
期刊论文
MEDCHEMCOMM, 2016
Shen, Qi
;
Zhang, Changsheng
;
Liu, Hongbo
;
Liu, Yuting
;
Cao, Junyue
;
Zhang, Xiaolin
;
Liang, Yuan
;
Zhao, Meiping
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
SMALL-MOLECULE INHIBITORS
TNF-ALPHA
FACTOR ANTAGONISTS
BINDING
OLIGOMERIZATION
SUPERFAMILY
RECEPTORS
DISCOVERY
DOMAIN
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