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4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
Tan, Li; Zhang, Zhang; Gao, Dongylin; Luo, Jinfeng; Tu, Zheng-Chao; Li, Zhengqiu; Peng, Lijie; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:23/0  |  提交时间:2016/12/16
4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
作者:  Tan, Li;  Zhang, Zhang;  Gao, Dongylin;  Luo, Jinfeng;  Tu, Zheng-Chao
收藏  |  浏览/下载:17/0  |  提交时间:2018/12/13
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:  Smaill, Jeff;  Lu, Xiaoyun;  Cheng, Huimin;  Zhang, Zhang;  Li, Yingjun
收藏  |  浏览/下载:48/0  |  提交时间:2018/12/13
Small Molecule Discoidin Domain Receptor Kinase Inhibitors and Potential Medical Applications 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 8, 页码: 3287-3301
作者:  Li, Yupeng;  Lu, Xiaoyun;  Ren, Xiaomei;  Ding, Ke
收藏  |  浏览/下载:15/0  |  提交时间:2018/12/13
N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 543-547
作者:  Ding, Ke;  Cheng, Huimin;  Zhang, Zhang;  Zhuang, Xiaoxi;  Li, Yingjun
收藏  |  浏览/下载:18/0  |  提交时间:2018/12/13
Small Molecule Discoidin Domain Receptor Kinase Inhibitors and Potential Medical Applications 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 8, 页码: 3287-3301
Li, Yupeng; Lu, Xiaoyun; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2016/12/16
N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 543-547
Li, Yingjun; Cheng, Huimin; Zhang, Zhang; Zhuang, Xiaoxi; Luo, Jinfeng; Long, Huoyou; Zhou, Yang; Xu, Yong; Taghipouran, Rana; Li, Dan; Patterson, Adam; Smaill, Jeff; Tu, Zhengchao; Wu, Donghai; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:17/0  |  提交时间:2016/12/16
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
作者:  Wang, Deping;  Feng, Yubing;  Zhuang, Xiaoxi;  Zhang, Fengxiang;  Liu, Jianqi
收藏  |  浏览/下载:23/0  |  提交时间:2018/12/13
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
Ren, Xiaomei; Pan, Xiaofen; Zhang, Zhang; Wang, Deping; Lu, Xiaoyun; Li, Yupeng; Wen, Donghai; Long, Huoyou; Luo, Jinfeng; Feng, Yubing; Zhuang, Xiaoxi; Zhang, Fengxiang; Liu, Jianqi; Leng, Fang; Lang, Xingfen; Bai, Yang; She, Miaoqin; Tu, Zhengchao; Pan, Jingxuan; Ding, Ke
收藏  |  浏览/下载:24/0  |  提交时间:2016/12/16


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