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Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
收藏  |  浏览/下载:85/0  |  提交时间:2020/12/24
Deep Learning Enhancing Kinome-Wide Polypharmacology Profiling: Model Construction and Experiment Validation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 16, 页码: 8723-8737
作者:  Li, Xutong;  Li, Zhaojun;  Wu, Xiaolong;  Xiong, Zhaoping;  Yang, Tianbiao
收藏  |  浏览/下载:28/0  |  提交时间:2020/12/21
Deep Learning Enhancing Kinome-Wide Polypharmacology Profiling: Model Construction and Experiment Validation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 16, 页码: 8723-8737
作者:  Li, Xutong;  Li, Zhaojun;  Wu, Xiaolong;  Xiong, Zhaoping;  Yang, Tianbiao
收藏  |  浏览/下载:23/0  |  提交时间:2020/12/21
Cryo-EM structure of an activated VIP1 receptor-G protein complex revealed by a NanoBiT tethering strategy 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  Duan, Jia;  Shen, Dan-dan;  Zhou, X. Edward;  Bi, Peng;  Liu, Qiu-feng
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/24
Sorting Nexin 10 Mediates Metabolic Reprogramming of Macrophages in Atherosclerosis Through the Lyn-Dependent TFEB Signaling Pathway 期刊论文
CIRCULATION RESEARCH, 2020, 卷号: 127, 期号: 4, 页码: 534-549
作者:  You, Yan;  Bao, Wei-Lian;  Zhang, Su-Lin;  Li, Hai-Dong;  Li, Hui
收藏  |  浏览/下载:48/0  |  提交时间:2020/12/24
Anti-hepatitis B virus activity of swertisin isolated from Iris tectorum Maxim 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2020, 卷号: 257, 页码: 9
作者:  Xu, Hong-Yan;  Ren, Ji-Hua;  Su, Yu;  Ren, Fang;  Zhou, Yu-Jiao
收藏  |  浏览/下载:25/0  |  提交时间:2020/12/24
Integrative Proteomic Characterization of Human Lung Adenocarcinoma 期刊论文
CELL, 2020, 卷号: 182, 期号: 1, 页码: 245-+
作者:  Xu, Jun-Yu;  Zhang, Chunchao;  Wang, Xiang;  Zhai, Linhui;  Ma, Yiming
收藏  |  浏览/下载:53/0  |  提交时间:2020/12/24
23,24-Dihydrocucurbitacin B promotes lipid clearance by dual transcriptional regulation of LDLR and PCSK9 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 327-335
作者:  Li, Hui-hui;  Li, Jun;  Zhang, Xian-jing;  Li, Jiao-meng;  Xi, Cong
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Identification and structural insight of an effective PPAR gamma modulator with improved therapeutic index for anti-diabetic drug discovery 期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 8, 页码: 2260-2268
作者:  Jiang, Haowen;  Zhou, X. Edward;  Shi, Jingjing;  Zhou, Zhi;  Zhao, Guanguan
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Diffuse large B-cell lymphoma with low F-18-fluorodeoxyglucose avidity features silent B-cell receptor signaling 期刊论文
LEUKEMIA & LYMPHOMA, 2020, 页码: 8
作者:  Sheng, Dong;  Li, Ting;  Wang, Wei-Ge;  Li, Meng-Jiao;  Jiang, Kai-Long
收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01


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