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科研机构
合肥物质科学研究院 [6]
安徽大学 [5]
大连理工大学 [1]
广州地球化学研究所 [1]
暨南大学 [1]
湖南大学 [1]
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期刊论文 [16]
发表日期
2018 [16]
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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2018, 卷号: 81, 期号: 11, 页码: 2531-2538
作者:
Wang, Qi
;
Hu, Zhenquan
;
Li, Xixiang
;
Wang, Aoli
;
Wu, Hong
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/25
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
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  |  
浏览/下载:68/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
Two new tricycloalternarenes from Hawaiian endophytic fungus Didymella sp FT433
期刊论文
TETRAHEDRON LETTERS, 2018, 卷号: 59, 期号: 36, 页码: 3381-3383
作者:
Li, Chunshun
;
Hu, Zhenquan
;
Liu, Qingsong
;
Wu, Xiaohua
;
Cao, Shugeng
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  |  
浏览/下载:31/0
  |  
提交时间:2019/11/11
Endophytic fungi
Didymella sp.
Tricycloalterene
Hawai'i
Bioactivity
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:
Liang, Xiaofei
;
Li, Feng
;
Chen, Cheng
;
Jiang, Zongru
;
Wang, Aoli
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/12/10
PI3K delta
Kinase inhibitor
Acute myeloid leukemia
Structure-activity relationship
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
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  |  
浏览/下载:64/0
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL
Hydrocarbon source for oil and gas indication associated with gas hydrate and its significance in the Qilian Mountain permafrost, Qinghai, Northwest China
期刊论文
MARINE AND PETROLEUM GEOLOGY, 2018, 卷号: 89, 页码: 202-215
作者:
Cheng, Bin
;
Xu, Jianbing
;
Lu, Zhenquan
;
Li, Yonghong
;
Wang, Weichao
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/08/19
Overcoming drug resistance with functional mesoporous titanium dioxide nanoparticles combining targeting, drug delivery and photodynamic therapy
期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2018, 卷号: 6, 页码: 7750-7759
作者:
Guo, Zhaoming
;
Zheng, Kun
;
Tan, Zhenquan
;
Liu, Ye
;
Zhao, Ziyin
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/02
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor
期刊论文
European Journal of Medicinal Chemistry, 2018, 卷号: Vol.156, 页码: 831-846
作者:
Zongru Jiang
;
Wenliang Wang
;
Fengming Zou
;
Jing Liu
;
Qingsong Liu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/04/22
PI3Kδ
Kinase
inhibitor
Acute
myeloid
leukemia
Structure-activity
relationship
Salviachinensines A–F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis
期刊论文
Journal of Natural Products, 2018, 卷号: Vol.81 No.11, 页码: 2531-2538
作者:
Xixiang Li
;
Qi Wang
;
Zhenquan Hu
;
Qingsong Liu
;
Jing Liu
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/04/24
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