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Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:  Liu, Xuesong;  Wang, Beilei;  Chen, Cheng;  Jiang, Zongru;  Hu, Chen
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/11
Salviachinensines A-F, Antiproliferative Phenolic Derivatives from the Chinese Medicinal Plant Salvia chinensis 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2018, 卷号: 81, 期号: 11, 页码: 2531-2538
作者:  Wang, Qi;  Hu, Zhenquan;  Li, Xixiang;  Wang, Aoli;  Wu, Hong
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/25
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming
收藏  |  浏览/下载:69/0  |  提交时间:2019/12/25
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:  Liang, Xiaofei;  Li, Feng;  Chen, Cheng;  Jiang, Zongru;  Wang, Aoli
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/10
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:  Wang, Qiang;  Liu, Feiyang;  Qi, Shuang;  Qi, Ziping;  Yan, Xiao-E.
收藏  |  浏览/下载:66/0  |  提交时间:2019/06/10
Hydrocarbon source for oil and gas indication associated with gas hydrate and its significance in the Qilian Mountain permafrost, Qinghai, Northwest China 期刊论文
MARINE AND PETROLEUM GEOLOGY, 2018, 卷号: 89, 页码: 202-215
作者:  Cheng, Bin;  Xu, Jianbing;  Lu, Zhenquan;  Li, Yonghong;  Wang, Weichao
收藏  |  浏览/下载:23/0  |  提交时间:2019/08/19
Fractional-Order Adaptive Backstepping Control of a Noncommensurate Fractional-Order Ferroresonance System 期刊论文
MATHEMATICAL PROBLEMS IN ENGINEERING, 2018
作者:  Wang, Yan;  Liu, Ling;  Liu, Chongxin;  Zhu, Ziwei;  Sun, Zhenquan
收藏  |  浏览/下载:12/0  |  提交时间:2019/11/19
Passive Acoustic Localization Based on COTS Mobile Devices 会议论文
2018 IEEE 24TH INTERNATIONAL CONFERENCE ON PARALLEL AND DISTRIBUTED SYSTEMS (ICPADS 2018), 2018-01-01
作者:  Liu, Tao;  Wang, Lei;  Qin, Zhenquan;  Qian, Chen;  Zhou, Xin
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/02
Enabling zigbee link performance robust under cross-technology interference 会议论文
13th International Conference on Wireless Algorithms, Systems, and Applications, WASA 2018, Tianjin, China, 2018-06-20
作者:  Sun, Yingxiao;  Qin, Zhenquan;  Hu, Junyu;  Wang, Lei;  Du, Jiaxin
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/02
Spoofing Attack Detection Using Physical Layer Information in Cross-Technology Communication 会议论文
2018 15TH ANNUAL IEEE INTERNATIONAL CONFERENCE ON SENSING, COMMUNICATION, AND NETWORKING (SECON), 2018-01-01
作者:  Lu, Bingxian;  Qin, Zhenquan;  Yang, Mingyi;  Xia, Xu;  Zhang, Renjie
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/02


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