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科研机构
上海药物研究所 [9]
内容类型
期刊论文 [9]
发表日期
2018 [9]
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发表日期:2018
内容类型:期刊论文
专题:上海药物研究所
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Artemisinin analogue SM934 ameliorates DSS-induced mouse ulcerative colitis via suppressing neutrophils and macrophages
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 10, 页码: 1633-1644
作者:
Yan, Yu-xi
;
Shao, Mei-juan
;
Qi, Qing
;
Xu, Yan-sheng
;
Yang, Xiao-qian
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
SM934
artemisinin analogue
ulcerative colitis
inflammatory bowel disease (IBD)
neutrophils macrophage
NF-kappa B
RAW 2647 cells
THP-1-derived macrophages
CUDC-907 displays potent antitumor activity against human pancreatic adenocarcinoma in vitro and in vivo through inhibition of HDAC6 to downregulate c-Myc expression
期刊论文
Acta pharmacologica Sinica, 2018
作者:
Fu, Xu-Hong
;
Zhang, Xiong
;
Yang, Hong
;
Xu, Xiao-Wei
;
Hu, Zong-Long
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Difuran-substituted quinoxalines as a novel class of PI3K alpha H1047R mutant inhibitors: Synthesis, biological evaluation and structure activity relationship
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 157, 页码: 37-49
作者:
Zhang, Ning
;
Yu, Zhimei
;
Yang, Xiaohong
;
Zhou, Yan
;
Tang, Qing
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Proliferation
Anticancer drug
Phosphatidylinositol 3-kinase inhibitor
Apoptosis
Structure-activity relationship
Acanthiline A, a pyrido[1,2-a]indole alkaloid from Chinese mangrove Acanthus ilicifolius
期刊论文
Journal of Asian natural products research, 2018, 页码: 1-5
作者:
Cai, You-Sheng
;
Sun, Ji-Zheng
;
Tang, Qing-Qing
;
Fan, Fengkai
;
Guo, Yue-Wei
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Topical administration of reversible SAHH inhibitor ameliorates imiquimod-induced psoriasis-like skin lesions in mice via suppression of TNF-alpha/IFN-gamma-induced inflammatory response in keratinocytes and T cell-derived IL-17
期刊论文
PHARMACOLOGICAL RESEARCH, 2018, 卷号: 129, 页码: 443-452
作者:
Lin, Ze-Min
;
Ma, Meng
;
Li, Heng
;
Qi, Qing
;
Liu, Yu-Ting
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Reversible S-adenosyl-L-homocysteine
hydrolase inhibitor
Keratinocyte
Inflammation
Interleukin-17
Imiquimod
Psoriasis
(5R)-5-hydroxytriptolide ameliorates anti-glomerular basement membrane glomerulonephritis in NZW mice by regulating Fc gamma receptor signaling
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 1, 页码: 107-116
作者:
Qi, Qing
;
Li, Heng
;
Lin, Ze-min
;
Yang, Xiao-qian
;
Zhu, Feng-hua
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
triptolide
(5R)-5-hydroxytriptolide (LLDT-8)
prednisolone
glomerulonephritis
immune complexes
inflammation
Fc gamma receptor signaling
artemisininanaloguesm934amelioratesdssinducedmouseulcerativecolitisviasuppressingneutrophilsandmacrophages
期刊论文
actapharmacologicasinica, 2018, 卷号: 39, 期号: 10, 页码: 1633
作者:
Yan Yuxi
;
Shao Meijuan
;
Qi Qing
;
Xu Yansheng
;
Yang Xiaoqian
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2020/07/01
NF-KAPPA-B
SODIUM-INDUCED COLITIS
MURINE COLITIS
MICE
CYTOKINES
CELLS
SM934
artemisinin analogue
ulcerative colitis
inflammatory bowel disease (IBD)
neutrophils macrophage
NF-kappa B
RAW 2647 cells
THP-1-derived macrophages
5r5hydroxytriptolideamelioratesantiglomerularbasementmembraneglomerulonephritisinnzwmicebyregulatingfcyreceptorsignaling
期刊论文
actapharmacologicasinica, 2018, 卷号: 39, 期号: 1, 页码: 107
作者:
Qi Qing
;
Li Heng
;
Lin Zemin
;
Yang Xiaoqian
;
Zhu Fenghua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/07/01
triptolide
(5R)-5-hydroxytriptolide (LLDT-8)
prednisolone
glomerulonephritis
immune complexes
inflammation
Fcy receptor signaling
(5R)-5-hydroxytriptolide ameliorates anti-glomerular basement membrane glomerulonephritis in NZW mice by regulating Fcy receptor signaling
期刊论文
Acta Pharmacologica Sinica, 2018, 卷号: 39, 期号: 1, 页码: 107
作者:
Qi Qing
;
Li Heng
;
Lin Zemin
;
Yang Xiaoqian
;
Zhu Fenghua
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/12/24
triptolide
(5R)-5-hydroxytriptolide (LLDT-8)
prednisolone
glomerulonephritis
immune complexes
inflammation
Fcy receptor signaling
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