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Discovery of a novel small inhibitor RJ19 targeting to human Hsp90 期刊论文
NUCLEAR SCIENCE AND TECHNIQUES, 2017, 卷号: 28, 期号: 10, 页码: -
作者:  Cao, HL;  Lyu, KK;  Liu, B;  Li, J;  He, JH
收藏  |  浏览/下载:20/0  |  提交时间:2018/08/30
Selenite-Induced Toxicity in Cancer Cells Is Mediated by Metabolic Generation of Endogenous Selenium Nanoparticles 期刊论文
JOURNAL OF PROTEOME RESEARCH, 2015, 卷号: 14, 期号: 2, 页码: 1127—1136
作者:  Bao, P;  Chen, Z;  Tai, RZ;  Shen, HM;  Martin, FL
收藏  |  浏览/下载:18/0  |  提交时间:2015/12/09
Multi-substituted 8-aminoimidazo[1,2-a]pyrazines by Groebke-Blackburn-Bienayme reaction and their Hsp90 inhibitory activity 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2015, 卷号: 13, 期号: 5, 页码: 1531—1535
作者:  Ren, J;  Yang, M;  Liu, HC;  Cao, DY;  Chen, DQ
收藏  |  浏览/下载:22/0  |  提交时间:2015/12/09
Identification of a new series of potent diphenol HSP90 inhibitors by fragment merging and structure-based optimization 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 11, 页码: 2525—2529
Ren, J; Li, J; Wang, YQ; Chen, WY; Shen, AJ; Liu, HC; Chen, DQ; Cao, DY; Li, YL; Zhang, NX; Xu, YC; Geng, MY; He, JH; Xiong, B; Shen, JK
收藏  |  浏览/下载:39/0  |  提交时间:2015/03/13
Structure insights into mechanisms of ATP hydrolysis and the activation of human heat-shock protein 90 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2012, 卷号: 44, 期号: 4, 页码: 300
Li, Jian(李健); Sun, Lihua(孙丽华); Xu, Chunyan(徐春艳); Yu, Feng(郁峰); Zhou, Huan; Zhao, Yanlong; Zhang, Jian; Cai, Jianhua; Mao, Cheney; Tang, Lin(唐琳); Xu, Yechun; He, Jianhua(何建华)
收藏  |  浏览/下载:17/0  |  提交时间:2013/09/11
Crystal Structures of N-terminal Domain of Human Hsp90 With ATP Analogues Reveal The Functional Regulation of Hsp90 期刊论文
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2012, 卷号: 39, 期号: 10
Li, J(李健); Sun, LH(孙丽华); Xu, CY(徐春艳); Yu, F(郁峰); Zhou, H(周欢); Tang, L(唐琳); He, JH(何建华)
收藏  |  浏览/下载:19/0  |  提交时间:2013/09/11


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