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Discovery of Cyclic Peptidomimetic Ligands Targeting the Extracellular Domain of EGFR 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 11219-11228
作者:  Zheng, Mengmeng;  Li, Chunpu;  Zhou, Mi;  Jia, Ru;  Cai, Gang
收藏  |  浏览/下载:68/0  |  提交时间:2021/11/04
A novel tricyclic BTK inhibitor suppresses B cell responses and osteoclastic bone erosion in rheumatoid arthritis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:  Liu, Yu-ting;  Ding, Hui-hua;  Lin, Ze-min;  Wang, Que;  Chen, Li
收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
收藏  |  浏览/下载:87/0  |  提交时间:2020/12/24
DW14006 as a direct AMPK alpha 1 activator improves pathology of AD model mice by regulating microglial phagocytosis and neuroinflammation 期刊论文
BRAIN BEHAVIOR AND IMMUNITY, 2020, 卷号: 90, 页码: 55-69
作者:  Lv, Jianlu;  Wang, Wei;  Zhu, Xialin;  Xu, Xiaoju;  Yan, Qiuying
收藏  |  浏览/下载:33/0  |  提交时间:2020/12/21
Exogenous FABP4 interferes with differentiation, promotes lipolysis and inflammation in adipocytes 期刊论文
ENDOCRINE, 2020, 卷号: 67, 期号: 3, 页码: 587-596
作者:  Dou, Hui-Xia;  Wang, Ting;  Su, Hai-Xia;  Gao, Ding-Ding;  Xu, Ye-Chun
收藏  |  浏览/下载:48/0  |  提交时间:2020/07/01
Identification and structural insight of an effective PPAR gamma modulator with improved therapeutic index for anti-diabetic drug discovery 期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 8, 页码: 2260-2268
作者:  Jiang, Haowen;  Zhou, X. Edward;  Shi, Jingjing;  Zhou, Zhi;  Zhao, Guanguan
收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
A molecular switch regulating transcriptional repression and activation of PPAR gamma 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 14
作者:  Shang, Jinsai;  Mosure, Sarah A.;  Zheng, Jie;  Brust, Richard;  Bass, Jared
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/24
Designing of novel ERR gamma inverse agonists by molecular modeling studies of docking and 3D-QSAR on hydroxytamoxifen derivatives 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2019, 卷号: 28, 期号: 10, 页码: 1661-1673
作者:  Li, Rui;  Du, Yongli;  Shen, Jingkang
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Discovery of betulinaldehyde as a natural ROR gamma t agonist 期刊论文
FITOTERAPIA, 2019, 卷号: 137, 页码: 8
作者:  Yang, Feng;  Zhang, Ruihan;  Ni, Dongxuan;  Luo, Xiaomin;  Chen, Shijie
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Xanthatin inhibits STAT3 and NF-kappa B signalling by covalently binding to JAK and IKK kinases 期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2019, 卷号: 23, 期号: 6, 页码: 4301-4312
作者:  Liu, Man;  Xiao, Cheng-qian;  Sun, Ming-wei;  Tan, Min-jia;  Hu, Li-hong
收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01


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