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科研机构
上海药物研究所 [32]
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期刊论文 [31]
会议论文 [1]
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2021 [1]
2019 [2]
2018 [2]
2016 [9]
2015 [4]
2014 [2]
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HSP70-16 and VDAC3 jointly inhibit seed germination under cold stress in Arabidopsis
期刊论文
PLANT CELL AND ENVIRONMENT, 2021, 页码: 12
作者:
Ashraf, Muhammad
;
Mao, Qionglei
;
Hong, Jun
;
Shi, Lei
;
Ran, Xiaoruo
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2021/08/17
ABA transport
cold stress
heat shock protein
seed germination
voltage-dependent anion channel protein
Design, Synthesis and Pharmacological Evaluation of Novel Hsp90N-terminal Inhibitors Without Induction of Heat Shock Response
期刊论文
CHEMISTRYOPEN, 2019, 卷号: 8, 期号: 3, 页码: 344-353
作者:
Liu, Peng
;
Chen, Xiangling
;
Zhu, Jianming
;
Li, Bo
;
Chen, Zhaoqiang
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/07/01
autophagy
Hsp72
Hsp90 inhibitor
triazines
antitumor activity
Inhibition of HSP90 beta Improves Lipid Disorders by Promoting Mature SREBPs Degradation via the Ubiquitin-proteasome System
期刊论文
THERANOSTICS, 2019, 卷号: 9, 期号: 20, 页码: 5769-5783
作者:
Zheng, Zu-Guo
;
Zhang, Xin
;
Liu, Xiao-Xiao
;
Jin, Xiu-Xiu
;
Dai, Lunzhi
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
HSP90 beta
lipid metabolism
corylin
SREBPs
proteasomal degradation
Discovery of FS36 as a Novel Human Hsp90 Inhibitor
期刊论文
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2018, 卷号: 45, 期号: 7, 页码: 736-744
作者:
Li Gen
;
Lu Kai-Kai
;
Li Jian
;
Yin Xiu-Shan
;
Zhao Dong
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
heat shock protein 90
antitumor drugs
inhibitor
X-ray diffraction
complex crystal structure
Design, synthesis and pharmacological evaluation of ALK and Hsp90 dual inhibitors bearing resorcinol and 2,4-diaminopyrimidine motifs
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 76-86
作者:
Geng, Kaijun
;
Liu, Hongchun
;
Song, Zilan
;
Zhang, Chi
;
Zhang, Minmin
收藏
  |  
浏览/下载:180/0
  |  
提交时间:2019/01/08
Heat shock protein 90 (Hsp90)
Tyrosine kinase ALK
Dual inhibitor
Drug resistance
Antiproliferative activity
Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 12, 页码: 1587-1596
作者:
Wang, Yue-qin
;
Shen, Ai-jun
;
Sun, Jing-ya
;
Wang, Xin
;
Liu, Hong-chun
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
non-small cell lung cancer
gefitinib resistance
Hsp90
Senkyunolide I attenuates oxygen-glucose deprivation/reoxygenation-induced inflammation in microglial cells
期刊论文
BRAIN RESEARCH, 2016, 卷号: 1649, 页码: 123-131
作者:
Hu, Yang-ye
;
Wang, Yuan
;
Liang, Shuang
;
Yu, Xue-li
;
Zhang, Lei
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Senkyunolide I
Microglial cells
Oxygen-glucose deprivation/reoxygenation
TLR4/NF-kappa B pathway
HSF-1/Hsp70
Regulation of Ubiquitin-like with Plant Homeodomain and RING Finger Domain 1 (UHRF1) Protein Stability by Heat Shock Protein 90 Chaperone Machinery
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2016, 卷号: 291, 期号: 38, 页码: 20125-20135
作者:
Ding, Guangjin
;
Chen, Peilin
;
Zhang, Hui
;
Huang, Xiaojie
;
Zang, Yi
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
70-kilodalton heat shock protein (HSP70)
cancer therapy
DNA methylation
protein degradation
ubiquitin
Acid-Activatable Versatile Micelleplexes for PD-L1 Blockade Enhanced Cancer Photodynamic Immunotherapy
期刊论文
NANO LETTERS, 2016, 卷号: 16, 期号: 9, 页码: 5503-5513
作者:
Wang, Dangge
;
Wang, Tingting
;
Liu, Jianping
;
Yu, Haijun
;
Jiao, Shi
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Micelleplexes
acid-activatable
photodynamic therapy
cancer immunotherapy
RNA interference
Y-632 inhibits heat shock protein 90 (Hsp90) function by disrupting the interaction between Hsp90 and Hsp70/Hsp90 organizing protein, and exerts antitumor activity in vitro and in vivo
期刊论文
CANCER SCIENCE, 2016, 卷号: 107, 期号: 6, 页码: 782-790
作者:
Wang, Wenqian
;
Liu, Yang
;
Zhao, Zhixin
;
Xie, Chengying
;
Xu, Yongping
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Hop
Hsp90
imatinib resistance
thiol oxidation
Y-632
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