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A camptothecin-based, albumin-binding prodrug enhances efficacy and safety in vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 226, 页码: 11
作者:  Cheng, Zhiyang;  Huang, Ying;  Shen, Qianqian;  Zhao, Yangrong;  Wang, Lei
收藏  |  浏览/下载:87/0  |  提交时间:2021/11/04
Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Dong, Ying;  Tang, Bi-xi;  Wang, Qi;  Zhou, Li-wei;  Li, Cong
收藏  |  浏览/下载:79/0  |  提交时间:2022/01/04
Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11
作者:  Fan, Shijie;  Yue, Liyan;  Wan, Wei;  Zhang, Yuanyuan;  Zhang, Bidong
收藏  |  浏览/下载:81/0  |  提交时间:2021/12/16
Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2 期刊论文
CELL RESEARCH, 2021, 页码: 3
作者:  Xie, Yuanchao;  Yin, Wanchao;  Zhang, Yumin;  Shang, Weijuan;  Wang, Zhen
收藏  |  浏览/下载:110/0  |  提交时间:2021/11/04
Kynurenine derivative 3-HAA is an agonist ligand for transcription factor YY1 期刊论文
Journal of Hematology & Oncology, 2021, 卷号: 14, 期号: 1
作者:  Shi,Zhaopeng;  Gan,Guifang;  Xu,Xiang;  Zhang,Jieying;  Yuan,Yuan
收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
Construction of 2-alkynyl aza-spiro[4,5]indole scaffolds via sequential C-H activations for modular click chemistry libraries 期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:  Zhang, Jun;  Wang, Mengmeng;  Wang, Huiying;  Xu, Hui;  Chen, Junjie
收藏  |  浏览/下载:77/0  |  提交时间:2021/11/04
Triptolide analog LLDT-8 ameliorates psoriasis-like dermatitis in BALB/c mice via suppressing the IL-36 alpha signaling pathway 期刊论文
PHARMACOLOGICAL RESEARCH, 2021, 卷号: 169, 页码: 11
作者:  Qi, Qing;  Li, Qian;  Zhu, Hongwen;  Lu, Huimin;  Yang, Xiaoqian
收藏  |  浏览/下载:71/0  |  提交时间:2021/08/17
Metabolic Study of Stable Isotope Labeled Indolinone Derivative in Hepatocyte Cell by UPLC/Q TOF MS 期刊论文
JOURNAL OF THE AMERICAN SOCIETY FOR MASS SPECTROMETRY, 2021, 卷号: 32, 期号: 6, 页码: 1538-1544
作者:  Yang, Jixia;  Zhang, Gongzheng;  Wang, Zhaoyang;  Meng, Jian;  Wen, Hongliang
收藏  |  浏览/下载:19/0  |  提交时间:2021/12/16
In vitro studies of deferasirox derivatives as potential organelle-targeting traceable anti-cancer therapeutics 期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:  Steinbrueck, Axel;  Sedgwick, Adam C.;  Han, Hai-Hao;  Zhao, Michael Y.;  Sen, Sajal
收藏  |  浏览/下载:42/0  |  提交时间:2021/06/11
Discovery of a Pyrimidinedione Derivative as a Potent and Orally Bioavailable Axl Inhibitor 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 7, 页码: 3956-3975
作者:  Zhang, Hefeng;  Peng, Xia;  Dai, Yang;  Shao, Jingwei;  Ji, Yinchun
收藏  |  浏览/下载:16/0  |  提交时间:2021/06/11


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