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A camptothecin-based, albumin-binding prodrug enhances efficacy and safety in vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 226, 页码: 11
作者:  Cheng, Zhiyang;  Huang, Ying;  Shen, Qianqian;  Zhao, Yangrong;  Wang, Lei
收藏  |  浏览/下载:86/0  |  提交时间:2021/11/04
Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:  Wei, Dan;  Wang, Hanlin;  Zeng, Qinghe;  Wang, Wenjing;  Hao, Bingbing
收藏  |  浏览/下载:30/0  |  提交时间:2021/12/16
Stereo-selective synthesis of non-canonical gamma-hydroxy-alpha-amino acids by enzymatic carbon-carbon bond formation 期刊论文
CATALYSIS SCIENCE & TECHNOLOGY, 2021, 页码: 6
作者:  Zhang, Rui;  Tan, Jiamu;  Luo, Zhenzhen;  Dong, Haihong;  Ma, Ningshan
收藏  |  浏览/下载:17/0  |  提交时间:2021/12/01
Diversity-Oriented Chemoenzymatic Synthesis of Sulfated and Nonsulfated Core 2 O-GalNAc Glycans 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 15, 页码: 10819-10828
作者:  Xu, Zhuojia;  Deng, Yaqi;  Zhang, Zhumin;  Ma, Wenjing;  Li, Wanjin
收藏  |  浏览/下载:35/0  |  提交时间:2021/11/04
Spiro ent-Clerodane Dimers: Discovery and Green Approaches for a Scalable Biomimetic Synthesis 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 15, 页码: 5647-5651
作者:  Li, Xing-Ren;  Yan, Bing-Chao;  Hu, Kun;  He, Shijun;  Sun, Han-Dong
收藏  |  浏览/下载:27/0  |  提交时间:2021/11/04
Conformation-Controlled Hydrogen-Bond-Mediated Aglycone Delivery Method for alpha-Xylosylation 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 15, 页码: 9945-9960
作者:  Cai, Deqin;  Bian, Ya;  Wu, Shengjie;  Ding, Kan
收藏  |  浏览/下载:15/0  |  提交时间:2021/11/04
Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 17
作者:  Lin, Lin;  Lin, Guangyao;  Zhou, Qingtong;  Bathgate, Ross A. D.;  Gong, Grace Qun
收藏  |  浏览/下载:31/0  |  提交时间:2021/08/17
Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
(-)-Isoscopariusin A, a Naturally Occurring Immunosuppressive Meroditerpenoid: Structure Elucidation and Scalable Chemical Synthesis 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 10
作者:  Yan, Bing-Chao;  Zhou, Min;  Li, Jian;  Li, Xiao-Nian;  He, Shi-Jun
收藏  |  浏览/下载:55/0  |  提交时间:2021/05/24
Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyridazinone derivatives as covalent FGFR inhibitors 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 3, 页码: 781-794
作者:  Wu, Xiaowei;  Dai, Mengdi;  Cui, Rongrong;  Wang, Yulan;  Li, Chunpu
收藏  |  浏览/下载:47/0  |  提交时间:2021/05/24


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