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科研机构
上海药物研究所 [89]
内容类型
期刊论文 [87]
会议论文 [1]
学位论文 [1]
发表日期
2021 [2]
2020 [4]
2019 [4]
2018 [13]
2017 [12]
2016 [6]
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Oncology [1]
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Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5-b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8644-8665
作者:
Kong, Qidi
;
Pan, Wei
;
Xu, Heng
;
Xue, Yaru
;
Guo, Bin
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/08/17
Nosiheptide analogues as potential antibacterial agents via dehydroalanine region modifications: Semi-synthesis, antimicrobial activity and molecular docking study
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 31, 页码: 10
作者:
Fan, Yafei
;
Chen, Hangfei
;
Mu, Ning
;
Wang, Wengui
;
Zhu, Kongkai
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/05/24
Nosiheptide analogues
Semi-synthesis
Antimicrobial activity
Molecular docking
Design and synthesis of novel desfluoroquinolone-aminopyrimidine hybrids as potent anti-MRSA agents with low hERG activity
期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 103, 页码: 10
作者:
Song, Runzhe
;
Wang, Yue
;
Wang, Minghui
;
Gao, Ruixuan
;
Yang, Teng
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/12/24
Desfluoroquinolone
Aminopyrimidine
Hybrids
Anti-MRSA
hERG activity
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 198, 页码: 11
作者:
Wang, Zhi-Cheng
;
Wei, Bingyan
;
Pei, Fang-Ning
;
Yang, Teng
;
Tang, Jie
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  |  
浏览/下载:14/0
  |  
提交时间:2020/12/24
Capsaicin
Nitrothiophene
Multidrug-resistant S. aureus
Antibacterial agent
Design, Synthesis and Biological Evaluation of Bengamide Analogues as ClpP Activators
期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 5
作者:
Kong, Xue-Qing
;
Wei, Bing-Yan
;
Yu, Chen-Xi
;
Guan, Xiang-Na
;
Ma, Wei-Ping
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24
Discovery of synergistic activity of fluoroquinolones in combination with antimicrobial peptides against clinical polymyxin-resistant Pseudomonas aeruginosa DK2
期刊论文
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 2, 页码: 413-417
作者:
Zheng, Xinyu
;
Cao, Qiao
;
Cao, Qin
;
Mao, Fei
;
Li, Xiaokang
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/07/01
Polymyxin B
Pseudomonas aeruginosa
Fluoroquinolones
Synergy
Cystic fibrosis
Antimicrobial peptides
Synthesis and biological evaluation of tryptophan-derived rhodanine derivatives as PTP1B inhibitors and anti-bacterial agents
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 172, 页码: 163-173
作者:
Liu, Hongyan
;
Sun, Danwen
;
Du, Hang
;
Zheng, Changji
;
Li, Jingya
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  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
Tryptophan-derived rhodanine
PTP1B inhibitor
Anti-bacterial
SAR
Sulfonium, an Underestimated Moiety for Structural Modification, Alters the Antibacterial Profile of Vancomycin Against Multidrug-Resistant Bacteria
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2019, 卷号: 58, 期号: 20, 页码: 6678-6682
作者:
Guan, Dongliang
;
Chen, Feifei
;
Qiu, Yunguang
;
Jiang, Bofeng
;
Gong, Likun
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
antibacterial
multidrug-resistant bacteria
sulfonium
vancomycin
Design, Synthesis, and Biological Evaluation of Novel DNA Gyrase-Inhibiting Spiropyrimidinetriones as Potent Antibiotics for Treatment of Infections Caused by Multidrug-Resistant Gram-Positive Bacteria
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 2950-2973
作者:
Shi, Chenghui
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  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
Design, synthesis and evaluation of hybrid of tetrahydrocarbazole with 2,4-diaminopyrimidine scaffold as antibacterial agents
期刊论文
European journal of medicinal chemistry, 2019, 卷号: 162, 页码: 203-211
作者:
Su, Liqiang
;
Li, Jiahui
;
Zhou, Zhen
;
Huang, Dongxia
;
Zhang, Yuanjin
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  |  
浏览/下载:121/0
  |  
提交时间:2019/01/08
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