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Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 224, 页码: 14
作者:  He, Yu-Long;  Chen, Meng-Ting;  Wang, Ting;  Zhang, Ming-Ming;  Li, Ying-Xia
收藏  |  浏览/下载:64/0  |  提交时间:2021/11/04
Combined treatment with FABP4 inhibitor ameliorates rosiglitazone-induced liver steatosis in obese diabetic db/db mice 期刊论文
BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2021, 页码: 10
作者:  Chen, Meng-Ting;  Huang, Jun-Shang;  Gao, Ding-Ding;  Li, Ying-Xia;  Wang, He-Yao
收藏  |  浏览/下载:42/0  |  提交时间:2021/08/17
Quantitative proteomics reveals Shexiang Baoxin Pill exerts cardioprotective effects by preserving energy metabolism in a rat model of myocardial infarction 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2021, 卷号: 266, 页码: 10
作者:  Yu, Feng;  Yu, Yue;  Tian, Saisai;  Zhou, Yanting;  Chen, Xiangling
收藏  |  浏览/下载:36/0  |  提交时间:2021/05/24
Exploration of Fragment Binding Poses Leading to Efficient Discovery of Highly Potent and Orally Effective Inhibitors of FABP4 for Anti-inflammation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 8, 页码: 4090-4106
作者:  Su, Haixia;  Zou, Yi;  Chen, Guofeng;  Dou, Huixia;  Xie, Hang
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Exogenous FABP4 interferes with differentiation, promotes lipolysis and inflammation in adipocytes 期刊论文
ENDOCRINE, 2020, 卷号: 67, 期号: 3, 页码: 587-596
作者:  Dou, Hui-Xia;  Wang, Ting;  Su, Hai-Xia;  Gao, Ding-Ding;  Xu, Ye-Chun
收藏  |  浏览/下载:48/0  |  提交时间:2020/07/01
Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 19, 页码: 16
作者:  He, Yulong;  Dou, Huixia;  Gao, Dingding;  Wang, Ting;  Zhang, Mingming
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
From hit to lead: Structure-based discovery of naphthalene-1 sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 44-59
作者:  Gao, Ding-Ding;  Dou, Hui-Xia;  Su, Hai-Xia;  Zhang, Ming-Ming;  Wang, Ting
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Combined Virtual Screening and Substructure Search for Discovery of Novel FABP4 Inhibitors 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017, 卷号: 57, 期号: 9, 页码: 2329-2335
作者:  Cai, Haiyan;  Wang, Ting;  Yang, Zhuo;  Xu, Zhijian;  Wang, Guimin
收藏  |  浏览/下载:11/0  |  提交时间:2019/01/08
Novel fatty acid binding protein 4 (FABP4) inhibitors: Virtual screening, synthesis and crystal structure determination 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 90, 页码: 241-250
作者:  Cai, Haiyan;  Liu, Qiufeng;  Gao, Dingding;  Wang, Ting;  Chen, Tiantian
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
Binding Modes of Three Inhibitors 8CA, F8A and I4A to A-FABP Studied Based on Molecular Dynamics Simulation 期刊论文
PLOS ONE, 2014, 卷号: 9, 期号: 6
作者:  Chen, Jianzhong;  Wang, Jinan;  Zhu, Weiliang
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08


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