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科研机构
上海药物研究所 [35]
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期刊论文 [35]
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2021 [1]
2020 [1]
2017 [1]
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Discovery of potential small molecular SARS-CoV-2 entry blockers targeting the spike protein
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Wang, Lin
;
Wu, Yan
;
Yao, Sheng
;
Ge, Huan
;
Zhu, Ya
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2021/11/04
SARS-CoV-2
natural products
virtual screening
spike protein
protein-protein interaction modulators
Identify potent SARS-CoV-2 main protease inhibitors via accelerated free energy perturbation-based virtual screening of existing drugs
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 44, 页码: 27381-27387
作者:
Li, Zhe
;
Li, Xin
;
Huang, Yi-You
;
Wu, Yaoxing
;
Liu, Runduo
收藏
  |  
浏览/下载:76/0
  |  
提交时间:2020/12/24
virtual screening
SARS-CoV-2
drug repurposing
free energy perturbation
main protease
Host-guest kinetic interactions between HP-beta-cyclodextrin and drugs for prediction of bitter taste masking
期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2017, 卷号: 140, 页码: 232-238
作者:
Guo, Zhen
;
Wu, Fei
;
Singh, Vikramjeet
;
Guo, Tao
;
Ren, Xiaohong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Cyclodextrin
Kinetic parameters
Taste masking
Surface plasmon resonance imaging
Modeling
Prediction
HER2-targeted antibody drug conjugates for ovarian cancer therapy
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2016, 卷号: 93, 页码: 274-286
作者:
Jiang, Jing
;
Dong, Lihou
;
Wang, Lei
;
Wang, Ling
;
Zhang, Jing
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2019/01/08
Ovarian cancer
Antibody drug conjugates (ADCs)
HER2/ErbB2
Monomethyl auristatin E (MMAE)
How Do Distance and Solvent Affect Halogen Bonding Involving Negatively Charged Donors?
期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2016, 卷号: 120, 期号: 34, 页码: 8784-8793
作者:
Chen, Zhaoqiang
;
Wang, Guimin
;
Xu, Zhijian
;
Wang, Jinan
;
Yu, Yuqi
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Generation and characterization of a human nanobody against VEGFR-2
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 6, 页码: 857-864
作者:
Ma, Lin
;
Gu, Kai
;
Zhang, Cheng-hai
;
Chen, Xue-tao
;
Jiang, Yi
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
nanobody
VEGFR2
anticancer agent
anti-angiogenesis
phage display
Simultaneous high-throughput determination of interaction kinetics for drugs and cyclodextrins by high performance affinity chromatography with mass spectrometry detection
期刊论文
ANALYTICA CHIMICA ACTA, 2016, 卷号: 909, 页码: 75-83
作者:
Wang, Caifen
;
Wang, Xiaobo
;
Xu, Xiaonan
;
Liu, Botao
;
Xu, Xu
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Cyclodextrin supramolecular systems
High performance affinity chromatography with mass spectrometry detection
High-throughput quantifying
Interactions kinetics
Stability and Characteristics of the Halogen Bonding Interaction in an Anion-Anion Complex: A Computational Chemistry Study
期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2016, 卷号: 120, 期号: 4, 页码: 610-620
作者:
Wang, Guimin
;
Chen, Zhaoqiang
;
Xu, Zhijian
;
Wang, Jinan
;
Yang, Yang
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Prediction of Rate Constant for Supramolecular Systems with Multiconfigurations
期刊论文
JOURNAL OF PHYSICAL CHEMISTRY A, 2016, 卷号: 120, 期号: 7, 页码: 981-991
作者:
Guo, Tao
;
Li, Haiyan
;
Wu, Li
;
Guo, Zhen
;
Yin, Xianzhen
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
Modified Release and Improved Stability of Unstable BCS II Drug by Using Cyclodextrin Complex as Carrier To Remotely Load Drug into Niosomes
期刊论文
MOLECULAR PHARMACEUTICS, 2016, 卷号: 13, 期号: 1, 页码: 113-124
作者:
Chi, Liandi
;
Wu, Delin
;
Li, Zhuo
;
Zhang, Minmin
;
Liu, Hongchun
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
niosomes
pseudolaric acid B
remote loading
pH gradient
retarded release
enzymatic stability
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