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科研机构
北京大学 [30]
内容类型
期刊论文 [29]
其他 [1]
发表日期
2017 [3]
2016 [5]
2015 [3]
2013 [2]
2012 [4]
2011 [2]
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专题:北京大学
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Antiamyloidogenic Activity of A beta 42-Binding Peptoid in Modulating Amyloid Oligomerization
期刊论文
SMALL, 2017
Zhao, Zijian
;
Zhu, Ling
;
Li, Haiyun
;
Cheng, Peng
;
Peng, Jiaxi
;
Yin, Yudan
;
Yang, Yang
;
Wang, Chen
;
Hu, Zhiyuan
;
Yang, Yanlian
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/04
aggregation,amyloid oligomerization,antiamyloidogenic,inhibitor,peptoids
GAMMA-SECRETASE INHIBITORS
SMALL-MOLECULE INHIBITORS
ALZHEIMERS-DISEASE
BETA-PEPTIDE
FIBRIL FORMATION
PROTEIN AGGREGATION
MOUSE MODEL
MECHANISM
NEUROTOXICITY
CONFORMATION
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
Tofacitinib ameliorates atherosclerosis and reduces foam cell formation in apoE deficient mice
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017
Wang, Zaicun
;
Wang, Shumei
;
Wang, Zunzhe
;
Yun, Tiantian
;
Wang, Chenchen
;
Wang, Huating
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/03
Tofacitinib
Atherosclerosis
Macrophage
Inflammation
Foam cell formation
PATHWAY-DEPENDENT MANNER
ABCA1 EXPRESSION
APOLIPOPROTEIN-E
JAK INHIBITOR
DIFFERENTIATION
MACROPHAGES
SUPPRESSORS
ACTIVATION
The cap-binding site of influenza virus protein PB2 as a drug target
期刊论文
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY, 2016
Severin, Chelsea
;
de Moura, Tales Rocha
;
Liu, Yong
;
Li, Keqin
;
Zheng, Xiaofeng
;
Luo, Ming
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
antiviral
inhibitor
drug design
broad spectrum
SUBUNIT
DOMAIN
1ST-IN-CLASS
INHIBITOR
MECHANISM
REVEALS
VX-787
STIM1 plays an important role in TGF-beta-induced suppression of breast cancer cell proliferation
期刊论文
ONCOTARGET, 2016
Cheng, Huanyi
;
Wang, Shiqiang
;
Feng, Renqing
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
TGF-beta
SOCE
STIM1
cell proliferation
breast cancer
PROMOTES TUMORIGENESIS
MESENCHYMAL TRANSITION
CALCIUM-CHANNELS
CRAC CHANNELS
CA2+ SENSOR
MCF-7 CELLS
STORE
MIGRATION
CYCLE
METASTASIS
Structure-based Inhibitor Design for the Intrinsically Disordered Protein c-Myc
期刊论文
SCIENTIFIC REPORTS, 2016
Yu, Chen
;
Niu, Xiaogang
;
Jin, Fan
;
Liu, Zhirong
;
Jin, Changwen
;
Lai, Luhua
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
SMALL-MOLECULE INHIBITOR
MYC/MAX DIMERIZATION
DRUG DESIGN
UNSTRUCTURED PROTEINS
SELECTIVE-INHIBITION
ACCURATE DOCKING
NMR-SPECTROSCOPY
LEUCINE-ZIPPER
BINDING
MODEL
Natural Product Kongensin A is a Non-Canonical HSP90 Inhibitor that Blocks RIP3-dependent Necroptosis
期刊论文
Cell Chemical Biology, 2016
Li, Dianrong
;
Li, Chao
;
Li, Lin
;
Chen, She
;
Wang, Lei
;
Li, Qiang
;
Wang, Xiaodong
;
Lei, Xiaoguang
;
Shen, Zhirong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
MIXED LINEAGE KINASE
DOMAIN-LIKE PROTEIN
CELL-DEATH
PROGRAMMED NECROSIS
BIOORTHOGONAL LIGATION
MOLECULAR CHAPERONE
RIP3
CANCER
MLKL
COMPLEX
6-C-(E-phenylethenyl)naringenin induces cell growth inhibition and cytoprotective autophagy in colon cancer cells
期刊论文
EUROPEAN JOURNAL OF CANCER, 2016
Zhao, Yueliang
;
Fan, Daming
;
Ru, Beibei
;
Cheng, Ka-Wing
;
Hu, Shuting
;
Zhang, Jiangwen
;
Li, Edmund T. S.
;
Wang, Mingfu
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2017/12/04
6-CEPN
Anticancer
Colon cancer
RAS
METHYLTRANSFERASE ACTIVITY
RAS
THERAPY
APOPTOSIS
DEATH
MODULATION
SIGNATURE
PATHWAYS
PROTEIN
ACID
Small-Molecule-Driven Direct Reprogramming of Mouse Fibroblasts into Functional Neurons
期刊论文
CELL STEM CELL, 2015
Li, Xiang
;
Zuo, Xiaohan
;
Jing, Junzhan
;
Ma, Yantao
;
Wang, Jiaming
;
Liu, Defang
;
Zhu, Jialiang
;
Du, Xiaomin
;
Xiong, Liang
;
Du, Yuanyuan
;
Xu, Jun
;
Xiao, Xiong
;
Wang, Jinlin
;
Chai, Zhen
;
Zhao, Yang
;
Deng, Hongkui
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
DOPAMINERGIC-NEURONS
CELL FATE
CONVERSION
PLURIPOTENCY
IDENTIFICATION
EXPRESSION
GENERATION
INHIBITORS
GENES
Ainsliadimer A selectively inhibits IKK alpha/beta by covalently binding a conserved cysteine
期刊论文
NATURE COMMUNICATIONS, 2015
Dong, Ting
;
Li, Chao
;
Wang, Xing
;
Dian, Longyang
;
Zhang, Xiuguo
;
Li, Lin
;
Chen, She
;
Cao, Ran
;
Li, Li
;
Huang, Niu
;
He, Sudan
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
NF-KAPPA-B
BIOMIMETIC SYNTHESES
ALLOSTERIC SITE
CANCER-THERAPY
BCL-X
ACTIVATION
PHOSPHORYLATION
INFLAMMATION
KINASE
UBIQUITINATION
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