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科研机构
北京大学 [21]
内容类型
期刊论文 [20]
其他 [1]
发表日期
2017 [5]
2016 [2]
2015 [2]
2014 [1]
2012 [1]
2011 [1]
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专题:北京大学
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Synthesis and evaluation of osimertinib derivatives as potent EGFR inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2017
Gao, Hongying
;
Yang, Zimo
;
Yang, Xinglin
;
Rao, Yu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
Osimertinib
N-Oxide metabolites
Fluoride
Non-small cell lung cancer
Epidermal growth factor receptor-tyrosine kinase inhibitors
CELL LUNG-CANCER
FACTOR RECEPTOR EGFR
MEDICINAL CHEMISTRY
TARGETED THERAPY
DRUG DISCOVERY
RESISTANCE
FLUORINE
MUTATIONS
MUTANT
PHARMACOKINETICS
Discovery of 2-((3-Acrylamido-4-methylphenyl)amino)-N-(2-methyl5-(3,4,5-trimethoxyben zamido)phenyI)-4-(methylamino)pyrimidine-5-carboxamide (CHMFL-BMX-078) as a Highly Potent and Selective Type II Irreversible Bone Marrow Kinase in the X Chro
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017
Liang, Xiaofei
;
Lv, Fengchao
;
Wang, Beilei
;
Yu, Kailin
;
Wu, Hong
;
Qi, Ziping
;
Jiang, Zongru
;
Chen, Cheng
;
Wang, Aoli
;
Miao, Weili
;
Wang, Wenchao
;
Hu, Zhenquan
;
Liu, Juan
;
Liu, Xiaochuan
;
Zhao, Zheng
;
Wang, Li
;
Zhang, Shanchuan
;
Ye, Zi
;
Wang, Chu
;
Ren, Tao
;
Wang, Yinsheng
;
Liu, Qingsong
;
Liu, Jing
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
GROWTH-FACTOR RECEPTOR
TYROSINE KINASE
COVALENT
ETK/BMX
FAMILY
CELLS
GENE
BTK
ACTIVATION
EXPRESSION
Designed inhibitor for nuclear localization signal of polo-like kinase 1 induces mitotic arrest
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2017
Chen, Fangjin
;
Zhuo, Xiaolong
;
Qin, Tan
;
Guo, Xiao
;
Zhang, Chuanmao
;
Lai, Luhua
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2017/12/03
anticancer
mitotic arrest
nuclear localization signal
Plk1 inhibitor
polo-like kinase 1
BOX DOMAIN
CANCER-THERAPY
CENTROSOME MATURATION
PLK1
PHOSPHORYLATION
AURORA
MITOSIS
ENTRY
Synthesis, crystal structure, enhanced photoluminescence properties and fluoride detection ability of S-heterocyclic annulated perylene diimide-polyhedral oligosilsesquioxane dye
期刊论文
JOURNAL OF MATERIALS CHEMISTRY C, 2017
Ben, Hai-Jie
;
Ren, Xiang-Kui
;
Song, Bo
;
Li, Xiaopeng
;
Feng, Yakai
;
Jiang, Wei
;
Chen, Er-Qiang
;
Wang, Zhaohui
;
Jiang, Shichun
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
AGGREGATION-INDUCED EMISSION
ORGANIC SOLAR-CELLS
PHYSICAL-PROPERTIES
SHAPE-PERSISTENT
LIQUID-CRYSTALS
SIDE-CHAINS
PERFORMANCE
BISIMIDE
POSS
SEMICONDUCTORS
A Combined DFT/IM-MS Study on the Reaction Mechanism of Cationic Ru(II)-Catalyzed Hydroboration of Alkynes
期刊论文
ACS CATALYSIS, 2017
Song, Li-Juan
;
Wang, Ting
;
Zhang, Xinhao
;
Chung, Lung Wa
;
Wu, Yun-Dong
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/03
hydroboration
hydrofunctionalization
trans-selectivity
ruthenium
density functional theory
mass spectrometry
MOBILITY-MASS-SPECTROMETRY
CATALYZED TRANS-HYDROBORATION
C-H ACTIVATION
GAS-PHASE
INTERNAL ALKYNES
TERMINAL ALKYNES
RUTHENIUM COMPLEXES
OXIDATIVE ADDITION
5+2 CYCLOADDITIONS
METAL-COMPLEXES
Discovery of Non-ATP-Competitive Inhibitors of Polo-like Kinase1
期刊论文
CHEMMEDCHEM, 2016
Yun, Taikangxiang
;
Qin, Tan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
inhibitors
kinase domain
non-ATP binding site
polo-like kinase1
virtual screening
1 PLK1 INHIBITORS
P38 MAP KINASE
CANCER-THERAPY
BINDING-SITE
BOX DOMAIN
PROTEIN
POLO-LIKE-KINASE-1
IDENTIFICATION
APOPTOSIS
DESIGN
Identification of acylthiourea derivatives as potent Plk1 PBD inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016
Yun, Taikangxiang
;
Qin, Tan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
Polo-like kinase 1
Polo-box domain
Small molecular inhibitor
Halogenosulfamoylphenyl acylthiourea
Binding affinity
In vitro assay
POLO-LIKE KINASE
INDUCE MITOTIC ARREST
BOX DOMAIN
PROGNOSTIC-SIGNIFICANCE
CANCER-CELLS
TUMOR-CELLS
DRUG DESIGN
EXPRESSION
DISCOVERY
DOCKING
Synthesis and properties of a novel Cu(II)-pyridineoxazoline containing polymeric catalyst for asymmetric Diels-Alder reaction
期刊论文
rsc advances, 2015
Wang, Heng
;
Li, Na
;
Yan, Zijia
;
Zhang, Jie
;
Wan, Xinhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/10
GOSTELI-CLAISEN REARRANGEMENT
OXAZOLINE-CONTAINING LIGANDS
BIS(OXAZOLINE) LIGANDS
ENANTIOSELECTIVE CATALYSIS
CHIRAL BIS(OXAZOLINE)
METHYLENE SPACER
TRANSITION-STATE
HIGH-PRESSURE
ALDEHYDES
IMMOBILIZATION
Base promoted hydrogenolysis of lignin model compounds and organosolv lignin over metal catalysts in water
期刊论文
chemical engineering science, 2015
Konnerth, Hannelore
;
Zhang, Jiaguang
;
Ma, Ding
;
Prechtl, Martin H. G.
;
Yan, Ning
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/11
Bimetallic nanoparticles
Base
Hydrogenolysis
Lignin
Biomass
HETEROGENEOUS NICKEL-CATALYSTS
ACIDIC IONIC LIQUIDS
RHODIUM-ON-CHARCOAL
ARYL ETHERS
WOOD LIGNIN
LIGNOCELLULOSIC BIOMASS
RENEWABLE CHEMICALS
ARENE HYDROGENATION
AQUEOUS-PHASE
CONVERSION
Exploring the Formation and Recognition of an Important G-Quadruplex in a HIF1 alpha Promoter and Its Transcriptional Inhibition by a Benzo[c]phenanthridine Derivative
期刊论文
journal of the american chemical society, 2014
Chen, Han
;
Long, Haitao
;
Cui, Xiaojie
;
Zhou, Jiang
;
Xu, Ming
;
Yuan, Gu
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/10
INDUCIBLE FACTOR-I
CIRCULAR-DICHROISM
CANCER-THERAPY
MESSENGER-RNA
HYPOXIA
HIF-1
GENE
SITE
ANGIOGENESIS
SELECTIVITY
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