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科研机构
上海药物研究所 [22]
内容类型
期刊论文 [22]
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2021 [1]
2015 [1]
2012 [2]
2011 [1]
2010 [3]
2009 [2]
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Pharmacolo... [2]
Chemistry [1]
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内容类型:期刊论文
专题:上海药物研究所
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Discovery of SARS-CoV-2-E channel inhibitors as antiviral candidates
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 7
作者:
Wang, Yi
;
Fang, Sui
;
Wu, Yan
;
Cheng, Xi
;
Zhang, Lei-ke
收藏
  |  
浏览/下载:106/0
  |  
提交时间:2021/08/17
SARS-CoV-2
envelope protein (2-E)
cation channel
high-throughput screening (HTS)
anti-virus
TREK1 channel blockade induces an antidepressant-like response synergizing with 5-HT1A receptor signaling
期刊论文
EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2015, 卷号: 25, 期号: 12, 页码: 2426-2436
作者:
Ye, Dongqing
;
Li, Yang
;
Zhang, Xiangrong
;
Guo, Fei
;
Geng, Leiyu
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
TWIK-related mechano-gated K+ channel (TREK1)
Antidepressant
SID1900
5-HT1A receptor
Chronic unpredictable mild stress (CUMS)
Brain derived neurotrophic factor (BDNF)
Discovery of N-(3,5-bis(1-pyrrolidylmethyl)-4-hydroxybenzyl)-4-methoxybenzenesulfamide (sulcardine) as a novel anti-arrhythmic agent
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 9, 页码: 1176-1186
作者:
Bai, Dong-lu
;
Chen, Wei-zhou
;
Bo, Yun-xin
;
Dong, Yue-li
;
Kang, Ai-li
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
sulcardine
sulcardine sulfate
changrolin
heart
arrhythmias
aconitine
ouabain
sodium current
L-type calcium current
Comparison of the effects of DC031050, a class III antiarrhythmic agent, on hERG channel and three neuronal potassium channels
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 6, 页码: 728-736
作者:
Li, Ping
;
Sun, Hai-feng
;
Zhou, Ping-zheng
;
Ma, Chao-ying
;
Hu, Guo-yuan
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
dofetilide
DC031050
class III antiarrhythmic agent
hERG
KCNQ
Kv1.2
delayed rectifier potassium current
Acacetin causes a frequency- and use-dependent blockade of hKv1.5 channels by binding to the S6 domain
期刊论文
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2011, 卷号: 51, 期号: 6, 页码: 966-973
作者:
Wu, Hui-Jun
;
Wu, Wei
;
Sun, Hai-Ying
;
Qin, Guo-Wei
;
Wang, Hong-Bing
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Acacetin
hKv1.5
Tonic blockade
Open channel blockade
Rate-dependent blockade
Tetrahydroberberine blocks ATP-sensitive potassium channels in dopamine neurons acutely-dissociated from rat substantia nigra pars compacta
期刊论文
NEUROPHARMACOLOGY, 2010, 卷号: 59, 期号: 7-8, 页码: 567-572
作者:
Wu, Chen
;
Yang, Kechun
;
Liu, Qiang
;
Wakui, Matoko
;
Jin, Guo-Zhang
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Tetrahydroberberine
Dopaminergic neurons
Substantia nigra compacta
ATP-sensitive K+ channel
Rotenone
Parch-clamp
State-dependent blockade of human ether-a-go-go-related gene (hERG) K+ channels by changrolin in stably transfected HEK293 cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2010, 卷号: 31, 期号: 8, 页码: 915-922
作者:
Chen, Wei-hai
;
Wang, Wen-yi
;
Zhang, Jie
;
Yang, Ding
;
Wang, Yi-ping
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
changrolin
human ether-a-go-go-related gene
torsades de pointes
whole-cell patch-clamp
anti-arrhythmic agent
State-dependent blockade of human ether-a-go-go-related gene (hERG) K~+ channels by changrolin in stably transfected HEK293 cells
期刊论文
Acta Pharmacologica Sinica, 2010, 卷号: 31, 期号: 8, 页码: 915
作者:
Chen Weihai
;
Wang Wenyi
;
Zhang Jie
;
Yang Ding
;
Wang Yiping
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2020/07/01
TORSADES-DE-POINTES
POTASSIUM CHANNELS
PROLONGATION
DERIVATIVES
BINDING
DRUGS
Arylbenzazepines Are Potent Modulators for the Delayed Rectifier K+ Channel: A Potential Mechanism for Their Neuroprotective Effects
期刊论文
PLOS ONE, 2009, 卷号: 4, 期号: 6
作者:
Chen, Xue-Qin
;
Zhang, Jing
;
Neumeyer, John L.
;
Jin, Guo-Zhang
;
Hu, Guo-Yuan
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
Current Strategies for the Discovery of K+ Channel Modulators
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2009, 卷号: 9, 期号: 4, 页码: 348-361
作者:
Ye, Deju
;
Wang, Jiang
;
Yu, Kunqian
;
Zhou, Yu
;
Jiang, Hualiang
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
Potassium channels
modulator
blocker
opener
virtual screening
chemistry strategy
MAOS
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