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Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 13, 页码: 2871-2881
Qin, Xuemei; Li, Zhipeng; Yang, Leifu; Liu, Peng; Hu, Liming; Zeng, Chengchu; Pan, Zhiyong
收藏  |  浏览/下载:59/0  |  提交时间:2016/12/16
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 6, 页码: 1571-1575
作者:  Lv, Yongjuan;  Qin, Xuemei;  Liu, Peng;  Li, Zhipeng;  Hu, Liming
收藏  |  浏览/下载:40/0  |  提交时间:2018/12/13
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 6, 页码: 1571-1575
Qin, Xuemei; Lv, Yongjuan; Liu, Peng; Li, Zhipeng; Hu, Liming; Zeng, Chengchu; Yang, Leifu
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 13, 页码: 2871-2881
作者:  Pan, Zhiyong;  Li, Zhipeng;  Yang, Leifu;  Liu, Peng;  Hu, Liming
收藏  |  浏览/下载:36/0  |  提交时间:2018/12/13
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:  Smaill, Jeff;  Lu, Xiaoyun;  Cheng, Huimin;  Zhang, Zhang;  Li, Yingjun
收藏  |  浏览/下载:48/0  |  提交时间:2018/12/13
C5-substituted pyrido[2,3-d]pyrimidin-7-ones as highly specific kinase inhibitors targeting the clinical resistance-related EGFR(T790M) mutant 期刊论文
MEDCHEMCOMM, 2015, 卷号: 6, 期号: 9, 页码: 1693-1697
作者:  Ding, Ke;  Ren, Xiaomei;  Zhang, Lianwen;  Yu, Lei;  Luo, Jinfeng
收藏  |  浏览/下载:47/0  |  提交时间:2018/12/13
C5-substituted pyrido[2,3-d]pyrimidin-7-ones as highly specific kinase inhibitors targeting the clinical resistance-related EGFR(T790M) mutant 期刊论文
MEDCHEMCOMM, 2015, 卷号: 6, 期号: 9, 页码: 1693-1697
Xu, Tianfeng; Peng, Ting; Ren, Xiaomei; Zhang, Lianwen; Yu, Lei; Luo, Jinfeng; Zhang, Zhang; Tu, Zhengchao; Tong, Linjiang; Huang, Zhaoru; Lu, Xiaoyun; Geng, Meiyu; Xie, Hua; Ding, Jian; Ding, Ke
收藏  |  浏览/下载:62/0  |  提交时间:2016/12/16
Synthesis and evaluation of 2-anilinopyrimidines bearing 3-aminopropamides as potential epidermal growth factor receptor inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 77, 期号: 1, 页码: 75-83
作者:  Han, C;  Wan, LD;  Ji, HB;  Ding, K;  Huang, ZJ
收藏  |  浏览/下载:27/0  |  提交时间:2015/07/22
Novel Hybrids of (Phenylsulfonyl)furoxan and Anilinopyrimidine as Potent and Selective Epidermal Growth Factor Receptor Inhibitors for Intervention of Non-Small-Cell Lung Cancer 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 11, 页码: 4738-4748
作者:  Han, C;  Huang, ZJ;  Zheng, C;  Wan, LD;  Zhang, LW
收藏  |  浏览/下载:17/0  |  提交时间:2015/07/22


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