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上海药物研究所 [19]
合肥物质科学研究院 [4]
西北高原生物研究所 [2]
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新疆理化技术研究所 [1]
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期刊论文 [31]
发表日期
2021 [31]
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Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Li, Teng-teng
;
Peng, Cheng
;
Wang, Ji-qiu
;
Xu, Zhi-jian
;
Su, Ming-bo
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2022/01/18
DPP4
distal mutation
enzymatic activity
molecular dynamics simulation
structure-function mechanism
Acetone Sensor Based on FAIMS-MEMS
期刊论文
MICROMACHINES, 2021, 卷号: 12, 期号: 12, 页码: 21
作者:
Zhang, Junna
;
Lei, Cheng
;
Liang, Ting
;
Liu, Ruifang
;
Zhao, Zhujie
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/02/17
diabetes
FAIMS-MEMS
acetone
reproducibility
stability
Advanced glycation end products via skin autofluorescence as potential marker of carotid atherosclerosis in patients with type 2 diabetes
期刊论文
NUTRITION METABOLISM AND CARDIOVASCULAR DISEASES, 2021, 卷号: 31
作者:
Ying, Lingwen
;
Shen, Yun
;
Zhang, Yang
;
Wang, Yikun
;
Liu, Yong
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/01/10
Advanced glycation end products
Carotid atherosclerosis
Cardiovascular events
Non-invasive
Type 2 diabetes
Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site
期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:
Wang, Jiang
;
Yang, Dehua
;
Cheng, Xi
;
Yang, Linlin
;
Wang, Zhaohui
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  |  
浏览/下载:27/0
  |  
提交时间:2022/01/04
Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 224, 页码: 14
作者:
He, Yu-Long
;
Chen, Meng-Ting
;
Wang, Ting
;
Zhang, Ming-Ming
;
Li, Ying-Xia
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2021/11/04
Type 2 diabetes mellitus
Dual FABP4/5 inhibitors
Anti-lipolytic and anti-inflammatory effects
Metabolic stability
Anti-diabetic activities
Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel alpha-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 115, 页码: 17
作者:
Xie, Hong-Xu
;
Zhang, Juan
;
Li, Yue
;
Zhang, Jin-He
;
Liu, Shan-Kui
收藏
  |  
浏览/下载:69/0
  |  
提交时间:2021/11/04
Tetrahydrobenzo[b]thiophen-2-yl)urea
alpha-Glucosidase inhibitors
Non-competitive inhibitor
Molecular docking
Anti-hyperglycaemic activity
Type 2 diabetes
Effects of Food on the Pharmacokinetic Properties and Mass Balance of Henagliflozin in Healthy Male Volunteers
期刊论文
CLINICAL THERAPEUTICS, 2021, 卷号: 43, 期号: 9, 页码: E264-E273
作者:
Chen, Zhen-dong
;
Chen, Qian
;
Zhu, Yun-ting
;
Zhang, Yi-fan
;
Zhan, Yan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/01/04
henagliflozin
food effects
mass balance
pharmacokinetics
SGLT-2 inhibitor
Signaling profiles in HEK 293T cells co-expressing GLP-1 and GIP receptors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 8
作者:
Wang, Yu-zhe
;
Yang, De-hua
;
Wang, Ming-wei
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/11/04
glucagon-like peptide-1 receptor
glucose-dependent insulinotropic peptide receptor
peptide 19
LY3298176
heteromerization
type 2 diabetes
Neo-clerodane Diterpenoids with Hypoglycemic Effects in Vivo from the Aerial Parts of Salvia hispanica L.
期刊论文
CHEMISTRY & BIODIVERSITY, 2021, 页码: 6
作者:
Fan, Min
;
Wang, Ting
;
Peng, Li-Yan
;
Huang, Jun-Shang
;
Wu, Xing-De
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/11/04
Salvia hispanica
neo-clerodane diterpenoid
salvihispin H
type 2 diabetes mellitus
Association of advanced glycation end products with diabetic retinopathy in type 2 diabetes mellitus
期刊论文
DIABETES RESEARCH AND CLINICAL PRACTICE, 2021, 卷号: 177
作者:
Ying, Lingwen
;
Shen, Yun
;
Zhang, Yang
;
Wang, Yikun
;
Liu, Yong
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/08/30
Diabetic retinopathy
Advanced glycation end products
Non-invasive
Type 2 diabetes
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