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科研机构
上海药物研究所 [8]
合肥物质科学研究院 [1]
内容类型
期刊论文 [9]
发表日期
2021 [9]
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New monoamine antidepressant, hypidone hydrochloride (YL-0919), enhances the excitability of medial prefrontal cortex in mice via a neural disinhibition mechanism
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Zhang, Yong-Mei
;
Ye, Lu-Yu
;
Li, Tian-Yu
;
Guo, Fan
;
Guo, Fei
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/01/04
YL-0919
medial prefrontal cortex
GABAergic neurons
5-HT1A receptor
GAD67-GFP transgenic mice
disinhibition
fluoxetine
electrophysiological recording
Anxiolytic effect of GABAergic neurons in the anterior cingulate cortex in a rat model of chronic inflammatory pain
期刊论文
MOLECULAR BRAIN, 2021, 卷号: 14, 期号: 1, 页码: 22
作者:
Shao, Fang-bing
;
Fang, Jun-fan
;
Wang, Si-si
;
Qiu, Meng-ting
;
Xi, Dan-ning
收藏
  |  
浏览/下载:113/0
  |  
提交时间:2021/11/04
Chronic inflammatory pain
Anxiety-like behavior
GABAergic system
Anterior cingulate cortex
synaptic transmission
Molecular insights into differentiated ligand recognition of the human parathyroid hormone receptor 2
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 32, 页码: 8
作者:
Wang, Xi
;
Cheng, Xi
;
Zhao, Lihua
;
Wang, Yuzhe
;
Ye, Chenyu
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/11/04
parathyroid hormone receptor 2
cryo-electron microscopy
G protein-coupled receptor
ligand recognition
syndromic short stature
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening
期刊论文
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:
Zhou, Qingtong
;
Guo, Wanjing
;
Dai, Antao
;
Cai, Xiaoqing
;
Vass, Marton
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/08/17
GLP-1R
virtual screening
allosteric modulator
drug discovery
molecular docking
TPN672: A Novel Serotonin-Dopamine Receptor Modulator for the Treatment of Schizophrenia
期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 378, 期号: 1, 页码: 20-30
作者:
Wang, Yu
;
He, Yang
;
Yang, Feipu
;
Abame, Melkamu Alemu
;
Wu, Chunhui
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/11/04
The Two Formyl Peptide Receptors Differently Regulate GPR84-Mediated Neutrophil NADPH Oxidase Activity
期刊论文
JOURNAL OF INNATE IMMUNITY, 2021, 页码: 15
作者:
Martensson, Jonas
;
Sundqvist, Martina
;
Manandhar, Asmita
;
Leremias, Loukas
;
Zhang, Linjie
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/05/24
Neutrophils
G protein-coupled receptors
Cross-talk
Nicotine adenine dinucleotide phosphate oxidase
Structures of the human dopamine D3 receptor-G(i) complexes
期刊论文
MOLECULAR CELL, 2021, 卷号: 81, 期号: 6, 页码: 1147-+
作者:
Xu, Peiyu
;
Huang, Sijie
;
Mao, Chunyou
;
Krumm, Brian E.
;
Zhou, X. Edward
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/05/24
CuO dot-decorated Cu@Gd2O3 core-shell hierarchical structure for Cu(i) self-supplying chemodynamic therapy in combination with MRI-guided photothermal synergistic therapy
期刊论文
MATERIALS HORIZONS, 2021, 卷号: 8
作者:
Zhang, Guilong
;
Xie, Wenteng
;
Xu, Zhaowei
;
Si, Yuanchun
;
Li, Qingdong
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/04/26
Sanguinarine is an agonist of TRPA1 channel
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2021, 卷号: 534, 页码: 226-232
作者:
Chi, Hao
;
Zhang, Xian
;
Chen, Xueqin
;
Fang, Sui
;
Ding, Qiang
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/05/24
Sanguinarine
Alkaloid
TRPA1
Agonist
Pain
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