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科研机构
上海药物研究所 [11]
近代物理研究所 [5]
海洋研究所 [2]
生态环境研究中心 [2]
合肥物质科学研究院 [2]
昆明植物研究所 [1]
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期刊论文 [24]
发表日期
2020 [24]
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Biochemist... [1]
Plant Scie... [1]
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DW14383 is an irreversible pan-FGFR inhibitor that suppresses FGFR-dependent tumor growth in vitro and in vivo
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:
Dai, Meng-di
;
Wang, Yue-liang
;
Fan, Jun
;
Dai, Yang
;
Ji, Yin-chun
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/05/24
receptor tyrosine kinase
FGFR inhibitor
DW14383
antitumor activity
Carbon Ion Therapy Inhibits Esophageal Squamous Cell Carcinoma Metastasis by Upregulating STAT3 Through the JAK2/STAT3 Signaling Pathway
期刊论文
FRONTIERS IN PUBLIC HEALTH, 2020, 卷号: 8, 页码: 11
作者:
Luo, Hongtao
;
Yang, Zhen
;
Zhang, Qiuning
;
Shao, Lihua
;
Wei, Shihong
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/12/13
carbon ion beam
esophageal squamous cell carcinoma
apoptosis
metastasis
JAK2
STAT3 pathway
The dual HDAC-PI3K inhibitor CUDC-907 displays single-agent activity and synergizes with PARP inhibitor olaparib in small cell lung cancer
期刊论文
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2020, 卷号: 39
作者:
Ma, Liying
;
Bian, Xing
;
Lin, Wenchu
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  |  
浏览/下载:40/0
  |  
提交时间:2020/11/30
SCLC
PI3K
HDAC
CUDC-907
PARP1
Olaparib
DSB repair
Combination treatment
NRF2 preserves genomic integrity by facilitating ATR activation and G2 cell cycle arrest
期刊论文
NUCLEIC ACIDS RESEARCH, 2020, 卷号: 48, 期号: 16, 页码: 9109-9123
作者:
Sun, Xiaohui
;
Wang, Yan
;
Ji, Kaihua
;
Liu, Yang
;
Kong, Yangyang
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/12/15
Radiosensitization of NSCLC cells to X-rays and carbon ions by the CHK1/CHK2 inhibitor AZD7762, Honokiol and Tunicamycin
期刊论文
RADIATION AND ENVIRONMENTAL BIOPHYSICS, 2020, 页码: 10
作者:
Liu, Bingtao
;
Chen, Weiqiang
;
Li, Hongbin
;
Li, Feifei
;
Jin, Xiaodong
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/12/15
Radiosensitivity
X-rays
Carbon ions
AZD7762
Honokiol
Tunicamycin
Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutation
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 16, 页码: 6
作者:
Su, Zhicheng
;
Yang, Tingyuan
;
Wang, Jie
;
Lai, Mengzhen
;
Tong, Linjiang
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/12/24
EGFR
NSCLC
C797S
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain
期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11
作者:
Chen, Yu
;
Bi, Xiaoyang
;
Zhang, Fengcai
;
Sun, Zhongya
;
Xu, Pan
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  |  
浏览/下载:24/0
  |  
提交时间:2020/12/24
In silico screening
Drug design
CBP
Bromodomain
Inhibitor
Acute Myeloblastic Leukemia
The effects of the Wnt/beta-catenin signaling pathway on apoptosis in HeLa cells induced by carbon ion irradiation
期刊论文
ONCOLOGY REPORTS, 2020, 卷号: 44, 期号: 1, 页码: 303-312
作者:
Si, Jing
;
Zhang, Jinhua
;
Gan, Lu
;
Gu, Menghuan
;
Xie, Yi
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/01/13
C-12(6+) irradiation
cervical cancer
Wnt/beta-catenin pathway
HLY78
radio-sensitivity
Protein Palmitoylation Regulates Cell Survival by Modulating XBP1 Activity in Glioblastoma Multiforme
期刊论文
MOLECULAR THERAPY-ONCOLYTICS, 2020, 卷号: 17
作者:
Chen, Xueran
;
Li, Hao
;
Fan, Xiaoqing
;
Zhao, Chenggang
;
Ye, Kaiqin
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/10/26
A novel M phase blocker, DCZ3301 enhances the sensitivity of bortezomib in resistant multiple myeloma through DNA damage and mitotic catastrophe
期刊论文
Journal of Experimental & Clinical Cancer Research, 2020, 卷号: 39, 期号: 1
作者:
Hu,Liangning
;
Li,Bo
;
Chen,Gege
;
Song,Dongliang
;
Xu,Zhijian
收藏
  |  
浏览/下载:95/0
  |  
提交时间:2020/07/01
Multiple myeloma
Drug-resistance
DNA damage response
Cell cycle
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