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Common activation mechanism of class A GPCRs 期刊论文
ELIFE, 2019, 卷号: 8, 页码: 31
作者:  Zhou, Qingtong;  Yang, Dehua;  Wu, Meng;  Guo, Yu;  Guo, Wangjing
收藏  |  浏览/下载:66/0  |  提交时间:2020/07/01
Colocalization Strategy Unveils an Underside Binding Site in the Transmembrane Domain of Smoothened Receptor 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 21, 页码: 9983-9989
作者:  Zhou, Fang;  Ding, Kang;  Zhou, Yiqing;  Liu, Yang;  Liu, Xiaoyan
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
TRAIL-based gene delivery and therapeutic strategies 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1373-1385
作者:  Zhong, Hui-hai;  Wang, Hui-yuan;  Li, Jian;  Huang, Yong-zhuo
收藏  |  浏览/下载:115/0  |  提交时间:2020/07/01
Designing of novel ERR gamma inverse agonists by molecular modeling studies of docking and 3D-QSAR on hydroxytamoxifen derivatives 期刊论文
MEDICINAL CHEMISTRY RESEARCH, 2019, 卷号: 28, 期号: 10, 页码: 1661-1673
作者:  Li, Rui;  Du, Yongli;  Shen, Jingkang
收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor 期刊论文
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 13, 页码: 8162-8169
作者:  Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Development of Small-Molecules Targeting Receptor Activator of Nuclear Factor-kappa B Ligand (RANKL)-Receptor Activator of Nuclear Factor-kappa B (RANK) Protein-Protein Interaction by Structure-Based Virtual Screening and Hit Optimization 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5370-5381
作者:  Jiang, Min;  Peng, Lei;  Yang, Kai;  Wang, Tianqi;  Yan, Xueming
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Ligand binding effects on the activation of the EGFR extracellular domain 期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2019, 卷号: 21, 期号: 15, 页码: 8141-8151
作者:  Shao, Qiang;  Zhu, Weiliang
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 3, 页码: 1373-1384
作者:  Chai, Hao;  Cheng, Xi;  Zhou, Bin;  Zhao, Lifen;  Lin, Xianhua
收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01
Human substance P receptor binding mode of the antagonist drug aprepitant by NMR and crystallography 期刊论文
NATURE COMMUNICATIONS, 2019, 卷号: 10, 页码: 8
作者:  Chen, Shuanghong;  Lu, Mengjie;  Liu, Dongsheng;  Yang, Lingyun;  Yi, Cuiying
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Structural basis for ligand recognition of the human thromboxane A(2) receptor 期刊论文
NATURE CHEMICAL BIOLOGY, 2019, 卷号: 15, 期号: 1, 页码: 27-+
作者:  Fan, Hengxin;  Chen, Shuanghong;  Yuan, Xiaojing;  Han, Shuo;  Zhang, Hui
收藏  |  浏览/下载:89/0  |  提交时间:2019/01/08


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