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科研机构
四川大学 [4]
上海药物研究所 [3]
西安交通大学 [2]
高能物理研究所 [1]
复旦大学上海医学院 [1]
湖南大学 [1]
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内容类型
期刊论文 [14]
发表日期
2018 [14]
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Multidisci... [1]
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发表日期:2018
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Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:
Hu, Jianping
;
Wang, Yingqing
;
Li, Yanlian
;
Cao, Danyan
;
Xu, Lin
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
BRD4
BI2536
Indoline
WPF binders
c-Myc
PD-L1
A cancer vaccine-mediated postoperative immunotherapy for recurrent and metastatic tumors
期刊论文
NATURE COMMUNICATIONS, 2018, 卷号: 9
作者:
Wang, Tingting
;
Wang, Dangge
;
Yu, Haijun
;
Feng, Bing
;
Zhou, Fangyuan
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
MGCD0103 induces apoptosis and simultaneously increases the expression of NF-kappa B and PD-L1 in classical Hodgkin's lymphoma
期刊论文
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2018, 卷号: 16, 期号: 5
作者:
Huang, Renhong
;
Zhang, Xiaowei
;
Min, Zhijun
;
Shadia, Abdelbari Sophia
;
Yang, Shun'e
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  |  
浏览/下载:3/0
  |  
提交时间:2019/12/05
Hodgkin's lymphoma
histone deacetylase inhibitor
nuclear factor-kappa B
programmed death-ligand 1
The risk of immune-related endocrine disorders associated with anti-PD-1 inhibitors therapy for solid tumors: A systematic review and meta-analysis
期刊论文
INTERNATIONAL IMMUNOPHARMACOLOGY, 2018, 卷号: 59, 页码: 328-338
作者:
Su, Qiang
;
Zhang, Xiao-chen
;
Wang, Di-ya
;
Zhang, Huai-rong
;
Zhu, Cheng
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/11/26
Immune-related endocrine disorders
PD-1 inhibitor
Meta-analysis
The efficacy and safety of anti-PD-1/PD-L1 antibody therapy versus docetaxel for pretreated advanced NSCLC: a meta-analysis
期刊论文
ONCOTARGET, 2018, 卷号: 9, 页码: 4239-4248
作者:
Huang, Guanghong
;
Sun, Xin
;
Liu, Dapeng
;
Zhang, Yunfeng
;
Zhang, Boxiang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/11/26
NSCLC
meta-analysis
PD-1/PD-L1
Immune checkpoint inhibitor
Dynamic change of pd-l1 expression on circulating tumor cells in advanced solid tumor patients undergoing pd-1 blockade therapy
期刊论文
Oncoimmunology, 2018, 卷号: 7, 期号: 7, 页码: 12
作者:
Yue, Chunyan
;
Jiang, Yubo
;
Li, Ping
;
Wang, Yuehua
;
Xue, Jian
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  |  
浏览/下载:84/0
  |  
提交时间:2019/04/23
Advanced solid tumor
Circulating tumor cells (ctcs)
Immunotherapy
Programmed death-ligand 1 (pd-l1)
Semi-quantitative analysis
Prognostic Factors for Checkpoint Inhibitor Based Immunotherapy: An Update With New Evidences
期刊论文
Frontiers in Pharmacology, 2018, 卷号: Vol.9
作者:
Xinyu Yan
;
Shouyue Zhang
;
Yun Deng
;
Peiqi Wang
;
Qianqian Hou
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/02/25
immunotherapy
checkpoint
inhibitor
PD-1
PD-L1
CTLA-4
Modulating the Tumor Microenvironment via Oncolytic Viruses and CSF-1R Inhibition Synergistically Enhances Anti-PD-1 Immunotherapy.
期刊论文
Molecular therapy : the journal of the American Society of Gene Therapy, 2018
作者:
Shi Gang
;
Yang Qianmei
;
Zhang Yujing
;
Jiang Qingyuan
;
Lin Yi
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/02/25
CSF-1R
inhibitor
anti-PD-1
antibody
combination
immunotherapy
oncolytic
virus
tumor
microenvironment
Modulating the Tumor Microenvironment via Oncolytic Viruses and CSF-1R Inhibition Synergistically Enhances Anti-PD-1 Immunotherapy.
期刊论文
Molecular therapy : the journal of the American Society of Gene Therapy, 2018
作者:
Shi Gang
;
Yang Qianmei
;
Zhang Yujing
;
Jiang Qingyuan
;
Lin Yi
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/02/25
CSF-1R
inhibitor
anti-PD-1
antibody
combination
immunotherapy
oncolytic
virus
tumor
microenvironment
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