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Identification of a cellularly active SIRT6 allosteric activator 期刊论文
NATURE CHEMICAL BIOLOGY, 2018, 卷号: 14, 期号: 12, 页码: 1118-+
作者:  Huang, Zhimin;  Zhao, Junxing;  Deng, Wei;  Chen, Yingyi;  Shang, Jialin
收藏  |  浏览/下载:95/0  |  提交时间:2019/01/08
Pharmacological characterization of hetrombopag, a novel orally active human thrombopoietin receptor agonist 期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2018, 卷号: 22, 期号: 11, 页码: 5367-5377
作者:  Xie, Chengying;  Zhao, Huajun;  Bao, Xubin;  Fu, Haoyu;  Lou, Liguang
收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming
收藏  |  浏览/下载:70/0  |  提交时间:2019/12/25
Emodin induces apoptosis in human hepatocellular carcinoma HepaRG cells via the mitochondrial caspase‑dependent pathway 期刊论文
Oncology reports, 2018, 卷号: 40, 期号: 4, 页码: 1985-1993
作者:  Dong, Xiaoxv;  Ni, Boran;  Fu, Jing;  Yin, Xingbin;  You, Longtai
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
DCZ3301, a novel aryl-guanidino inhibitor, induces cell apoptosis and cell cycle arrest via suppressing the PI3K/AKT pathway in T-cell leukemia/lymphoma 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2018, 卷号: 50, 期号: 7, 页码: 643-650
作者:  Xiao, Wenqin;  Li, Bo;  Sun, Xi;  Yu, Dandan;  Xie, Yongsheng
收藏  |  浏览/下载:87/0  |  提交时间:2019/01/08
Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors 期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 6
作者:  Wu, Yi-Zhe;  Ying, Hua-Zhou;  Xu, Lei;  Cheng, Gang;  Chen, Jing
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
The cyclin-dependent kinase 2 (CDK2) mediates hematopoiesis through G1-to-S transition in Chinese mitten crab Eriocheir sinensis 期刊论文
DEVELOPMENTAL AND COMPARATIVE IMMUNOLOGY, 2018, 卷号: 81, 页码: 156-166
作者:  Yang, Bin;  Jia, Yunke;  Jia, Zhihao;  Wang, Weilin;  Song, Xiaorui
收藏  |  浏览/下载:27/0  |  提交时间:2019/08/21
Constituents of Mediterranean Spices Counteracting Vascular Smooth Muscle Cell Proliferation: Identification and Characterization of Rosmarinic Acid Methyl Ester as a Novel Inhibitor 期刊论文
MOLECULAR NUTRITION & FOOD RESEARCH, 2018, 卷号: 62, 期号: 7
作者:  Liu, Rongxia;  Heiss, Elke H.;  Waltenberger, Birgit;  Blazevic, Tina;  Schachner, Daniel
收藏  |  浏览/下载:56/0  |  提交时间:2019/01/08
Lipid-Based Liquid Crystalline Nanoparticles Facilitate Cytosolic Delivery of siRNA via Structural Transformation 期刊论文
NANO LETTERS, 2018, 卷号: 18, 期号: 4, 页码: 2411-2419
作者:  He, Shufang;  Fan, Weiwei;  Wu, Na;  Zhu, Jingjing;  Miao, Yunqiu
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
A Novel Bromophenol Derivative BOS-102 Induces Cell Cycle Arrest and Apoptosis in Human A549 Lung Cancer Cells via ROS-Mediated PI3K/Akt and the MAPK Signaling Pathway 期刊论文
MARINE DRUGS, 2018, 卷号: 16, 期号: 2, 页码: 13
作者:  Guo, Chuan-Long;  Wang, Li-Jun;  Zhao, Yue;  Liu, Hua;  Li, Xiang-Qian
收藏  |  浏览/下载:24/0  |  提交时间:2019/08/21


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