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科研机构
上海药物研究所 [4]
山东大学 [3]
大连化学物理研究所 [1]
武汉轻工大学 [1]
中国医学科学院 北京... [1]
内容类型
期刊论文 [10]
发表日期
2018 [10]
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发表日期:2018
内容类型:期刊论文
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Metabolism and disposition of pyrotinib in healthy male volunteers: covalent binding with human plasma protein
期刊论文
Acta pharmacologica Sinica, 2018
作者:
Meng, Jian
;
Liu, Xiao-Yun
;
Ma, Sheng
;
Zhang, Hua
;
Yu, Song-da
收藏
  |  
浏览/下载:100/0
  |  
提交时间:2019/01/08
Stable Cocrystals and Salts of the Antineoplastic Drug Apatinib with Improved Solubility in Aqueous Solution
期刊论文
CRYSTAL GROWTH & DESIGN, 2018, 卷号: 18, 期号: 8, 页码: 4701-4714
作者:
Zhu, Bin
;
Wang, Jian-Rong
;
Zhang, Qi
;
Li, Meiqi
;
Guo, Chunyang
收藏
  |  
浏览/下载:71/0
  |  
提交时间:2019/01/08
Acylated iridoid diglycosides from the cultivated endangered ornamental tree Gmelina hainanensis
期刊论文
PHYTOCHEMISTRY LETTERS, 2018, 卷号: 25, 页码: 17-21
作者:
Xiong, Juan
;
Wu, Xi-Ying
;
Wang, Pei-Pei
;
Lau, Choiwan
;
Fan, Hui
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
Gmelina hainanensis
Endangered plant
Acylated iridoid glycosides
PTP1B inhibition
Recent advances in methods for the analysis of protein o-glycosylation at proteome level
期刊论文
JOURNAL OF SEPARATION SCIENCE, 2018, 卷号: 41, 期号: 1, 页码: 248-261
作者:
You, Xin
;
Qin, Hongqiang
;
Ye, Mingliang
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/06/20
Acetylgalactosamine
Acetylglucosamine
Enrichment Methods
Glycosylation
Proteomics
HLA and MuSK-positive myasthenia gravis: A systemic review and meta-analysis
期刊论文
ACTA NEUROLOGICA SCANDINAVICA, 2018, 卷号: 138, 期号: 3, 页码: 219-226
作者:
Hong, Y.
;
Li, H. -F.
;
Romi, F.
;
Skeie, G. O.
;
Gilhus, N. E.
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  |  
浏览/下载:4/0
  |  
提交时间:2019/12/11
genetic polymorphism
human leucocyte antigen
meta-analysis
muscle-specific tyrosine kinase
myasthenia gravis
Computational Strategy for Bound State Structure Prediction in Structure-Based Virtual Screening: A Case Study of Protein Tyrosine Phosphatase Receptor Type O Inhibitors
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2018, 卷号: 58, 期号: 11, 页码: 2331-2342
作者:
Hou, Xuben
;
Rooklin, David
;
Yang, Duxiao
;
Liang, Xiao
;
Li, Kangshuai
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/11
Specific effects of neuregulin-1β on the communication between DRG neurons and skeletal muscle cells in vitro
期刊论文
Journal of Muscle Research and Cell Motility, 2018
作者:
Cong M.
;
Li J.
;
Qiao Y.
;
Jing R.
;
Li H.
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/11
Dorsal root ganglion
Neuregulin-1β
Neuron
Signaling pathway
Skeletal muscle cell
Tyrosine kinase receptor
MicroRNA-208a Correlates Apoptosis and Oxidative Stress Induced by H2O2 through Protein Tyrosine Kinase/Phosphatase Balance in Cardiomyocytes
期刊论文
2018, 卷号: 59, 期号: 4, 页码: 829-836
作者:
Liu, Aijun
;
Sun, Yiping
;
Yu, Bo
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  |  
浏览/下载:3/0
  |  
提交时间:2020/01/03
Reactive oxygen species
Ischemia/reperfusion
non-encoding RNAs
PTPRG
PTPN4
Dietary supplementation of A-type procyanidins from litchi pericarp improves glucose homeostasis by modulating mTOR signaling and oxidative stress in diabetic ICR mice
期刊论文
Journal of Functional Foods, 2018, 卷号: 44, 页码: 155-165
作者:
Li, Xiaopeng
;
Wu, Qian
;
Sui, Yong
;
Li, Shuyi
;
Xie, Bijun
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/12/27
A-type procyanidins
Oxidative stress
Glucose homeostasis
Type 2 diabetes
mTOR
ACC1
acetyl coenzyme A carboxylase 1
ACL
ATP-citrate lyase
ALT
alanine aminotransferase
AST
aspartate aminotransferase
AUC
area under curve
BAT
brown adipose tissue
FAS
fatty acid synthase
FFA
free fatty acid
FoxO3a
Forkhead box O3a
FoxO1a
Forkhead box O3a
PKCβ
protein kinase C β
mTOR
mechanistic target of rapamycin
HDL
high-density lipoprotein
GHbA1c
glycated hemoglobin A1c
GK
glucokinase
G-6-Pase
glucose-6-phosphatase
GLP-1
glucagon-like peptide-1
GSH-PX
total glutathione peroxidase
HOMA-IR
homeostatic model assessment of insulin resistance
LDHA
lactate dehydrogenase
LDL
low-density lipoprotein
LPOPC
oligomeric procyanidins of litchi pericarp
MDA
malondialdehyde
MnSOD
manganese superoxide dismutase
mTOR
mechanistic target of rapamycin
OGTT
oral glucose tolerance test
PDH
pyruvate dehydrogenase
PEPCK
phosphoenolpyruvate carboxykinase
PFK
phosphofructokinase
PK
pyruvate kinase
PKCβ
protein kinase C β
PPG
postprandial blood glucose
S6K1
S6 Kinase 1
PKCβ
protein kinase C β
RTK
receptor tyrosine kinase
SREBP-1c
sterol regulatory element-binding protein 1c
ACL
ATP-citrate lyase
ACC1
acetyl coenzyme A carboxylase 1
FAS
fatty acid synthase
SCD1
stearoyl CoA desaturase 1
STZ
streptozotocin
S6K1
S6 kinase 1
PPG
postprandial blood glucose
ROS
reactive oxygen species
TC
total cholesterol
TG
triacylglycerol
STZ
streptozotocin
T-AOC
total antioxidant capacity
T-SOD
total superoxide dismutase
UCP-1
uncoupling protein 1
WAT
white adipose tissue
XOS
xylo-oligosaccharides
Synthesis and Biological Activities of Novel 2-Aminobenzimidazoles EGFR~(T790M) Inhibitors
期刊论文
Chinese Journal of Synthetic Chemistry, 2018, 卷号: 26, 期号: 9, 页码: 637-646
作者:
Duan Jingyi
;
Zhang Yinyong
;
Qian Anran
;
Tong Linjiang
;
Xie Hua
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
1-fluoro-2-nitroarene
trans-4-aminocyclohexanol hydrochloride
2-aminobenzimidazole
EGFR~(T790M) inhibitor
synthesis
biological activity
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