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Mutation L1196M-induced conformational changes and the drug resistant mechanism of anaplastic lymphoma kinase studied by free energy perturbation and umbrella sampling 期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2017, 卷号: 19, 期号: 44, 页码: 30239-30248
作者:  Chen, Jianzhong;  Wang, Jinan;  Zhu, Weiliang
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
DCZ3301, a novel cytotoxic agent, inhibits proliferation in diffuse large B-cell lymphoma via the STAT3 pathway 期刊论文
CELL DEATH & DISEASE, 2017, 卷号: 8
作者:  Sun, Xi;  Li, Bo;  Xie, Bingqian;  Xu, Zhijian;  Chang, Gaomei
收藏  |  浏览/下载:64/0  |  提交时间:2019/01/08
Structure-activity relationship investigation for benzonaphthyridinone derivatives as novel potent Bruton's tyrosine kinase (BTK) irreversible inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 545-557
作者:  Wang, Beilei;  Deng, Yuanxin;  Chen, Yongfei;  Yu, Kailin;  Wang, Aoli
收藏  |  浏览/下载:43/0  |  提交时间:2018/08/16
Discovery of N-(3-(5-((3-acrylamido-4-(morpholine-4-carbonyl) phenyl)amino)-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl)-4-(tert-butyl)benzamide (CHMFL-BTK-01) as a highly selective irreversible Bruton's tyrosine kinase (BTK) inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 131, 页码: 107-125
作者:  Liang, Qianmao;  Chen, Yongfei;  Yu, Kailin;  Chen, Cheng;  Zhang, Shouxiang
收藏  |  浏览/下载:39/0  |  提交时间:2018/07/26
Marine-derived chromopeptide A, a novel class I HDAC inhibitor, suppresses human prostate cancer cell proliferation and migration 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 4, 页码: 551-560
作者:  Sun, Jing-ya;  Wang, Ji-dong;  Wang, Xin;  Liu, Hong-chun;  Zhang, Min-min
收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
Luteolin induces apoptosis in vitro through suppressing the MAPK and PI3K signaling pathways in gastric cancer 期刊论文
ONCOLOGY LETTERS, 2017, 卷号: 14, 期号: 2, 页码: 1993-2000
作者:  Lu, XY (Lu, Xueying);  Li, YH (Li, Yanhong);  Li, XB (Li, Xiaobo);  Aisa, HA (Aisa, Haji Akber)
收藏  |  浏览/下载:19/0  |  提交时间:2017/12/11
Altered expression of microRNA-98 in IL-1 beta-induced cartilage degradation and its role in chondrocyte apoptosis 期刊论文
MOLECULAR MEDICINE REPORTS, 2017, 卷号: 16, 期号: 3
作者:  Ma, Sha;  Wang, Jing;  Chen, Lingqing;  Jin, Song;  Lin, Jun
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/04
Early anthracycline-induced cardiotoxicity monitored by echocardiographic Doppler parameters combined with serum hs-cTnT 期刊论文
ECHOCARDIOGRAPHY-A JOURNAL OF CARDIOVASCULAR ULTRASOUND AND ALLIED TECHNIQUES, 2017, 卷号: 34, 期号: 11
作者:  Zhang, Chu-Jie;  Pei, Xiao-Li;  Song, Fei-Yan;  Guo, Ye;  Zhang, Qun-Ling
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/05
Altered expression of microRNA-98 in IL-1β-induced cartilage degradation and its role in chondrocyte apoptosis 期刊论文
Molecular Medicine Reports, 2017, 卷号: 16, 期号: 3
作者:  Wang, Jing[0];  Chen, Lingqing[1];  Jin, Song[2];  Lin, Jun[3];  Zheng, Hongmei[4]
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05
Toxicity study of oxalicumone A, derived from a marine-derived fungus Penicillium oxalicum, in cultured renal epithelial cells 期刊论文
MOLECULAR MEDICINE REPORTS, 2017, 卷号: 15, 期号: 5, 页码: 2611-2619
作者:  Shi, S;  Guo, KB;  Wang, XG;  Chen, H;  Min, JB
收藏  |  浏览/下载:26/0  |  提交时间:2017/09/08


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