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Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 140, 页码: 510-527
作者:  Chen, Lingfeng;  Fu, Weitao;  Feng, Chen;  Qu, Rong;  Tong, Linjiang
收藏  |  浏览/下载:57/0  |  提交时间:2019/01/08
Facile Synthesis of Novel Perfluorocarbon-Modulated 4-Anilinoquinazoline Analogues 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2017, 卷号: 35, 期号: 11, 页码: 1693-1700
作者:  Shi, Huiping;  Lai, Bonan;  Chen, Shizhen;  Zhou, Xin;  Nie, Jing
收藏  |  浏览/下载:66/0  |  提交时间:2018/11/05
Quantitative Proteomics Reveals the Regulatory Networks of Circular RNA CDR1as in Hepatocellular Carcinoma Cells 期刊论文
JOURNAL OF PROTEOME RESEARCH, 2017, 卷号: 16, 期号: 10, 页码: 3891-3902
作者:  Yang, Xue;  Xiong, Qian;  Wu, Ying;  Li, Siting;  Ge, Feng
收藏  |  浏览/下载:97/0  |  提交时间:2019/09/26
Single-molecule imaging reveals the stoichiometry change of epidermal growth factor receptor during transactivation by beta(2)-adrenergic receptor 期刊论文
SCIENCE CHINA-CHEMISTRY, 2017, 卷号: 60, 期号: 10, 页码: 1310-1317
作者:  Zhang, Mingliang;  He, Kangmin;  Wu, Jimin;  Li, Nan;  Yuan, Jinghe
收藏  |  浏览/下载:77/0  |  提交时间:2018/04/25
DCLAK11对非小细胞肺癌细胞HCC827的抗肿瘤作用 期刊论文
中国医院药学杂志, 2017, 卷号: 37, 期号: 19, 页码: 1914-1917
作者:  郭小彬;  刘红椿;  丁健
收藏  |  浏览/下载:44/0  |  提交时间:2019/01/08
Structure-Guided Design of C4-alkyl-1,4-dihydro-2H-pyrimido[4,5-d][1,3]oxazin-2-ones as Potent and Mutant-Selective Epidermal Growth Factor Receptor (EGFR) L858R/T790M Inhibitors 期刊论文
SCIENTIFIC REPORTS, 2017, 卷号: 7
作者:  Hao, Yongjia;  Lyu, Jiankun;  Qu, Rong;  Sun, Deheng;  Zhao, Zhenjiang
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Active targeting theranostic iron oxide nanoparticles for MRI and magnetic resonance-guided focused ultrasound ablation of lung cancer 期刊论文
BIOMATERIALS, 2017, 卷号: 127, 页码: 25-35
作者:  Wang, Zhongling;  Qiao, Ruirui;  Tang, Na;  Lu, Ziwei;  Wang, Han
收藏  |  浏览/下载:48/0  |  提交时间:2018/01/10
Chitosan oligosaccharide inhibits EGF-induced cell growth possibly through blockade of epidermal growth factor receptor/imitogen-activated protein kinase pathway 期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2017, 卷号: 98, 页码: 502-505
作者:  Xu, Qingsong;  Wang, Wenjing;  Yang, Wen;  Du, Yuguang;  Song, Linsheng
收藏  |  浏览/下载:33/0  |  提交时间:2017/05/17
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:  Wang, Aoli;  Li, Xixiang;  Wu, Hong;  Zou, Fengming;  Yan, Xiao-E
收藏  |  浏览/下载:35/0  |  提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:  Wang, Aoli;  Li, Xixiang;  Wu, Hong;  Zou, Fengming;  Yan, Xiao-E
收藏  |  浏览/下载:44/0  |  提交时间:2018/07/26


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