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An Efficient Novel Synthesis of 14-O-[(4-Amino-6-hydroxy-pyrimidine-2-yl)thioacetyl]Mutilin and the Antibacterial Evaluation 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2017, 卷号: 36, 期号: 9, 页码: 1433-1438
作者:  Yi Yun-Peng;  Xu Wen-Jun;  Huang Xin;  Liang Jian-Ping;  Shang Ruo-Feng
收藏  |  浏览/下载:12/0  |  提交时间:2019/11/15
Synthesis, Crystal Structure and Biological Evaluation of 14-O-[(2-chloroacetamide-6-aminopyrimidine-2-yl)thioacetyl] Mutilin 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2017, 卷号: 36, 页码: 1327-1333
作者:  Zhou Xiang;  Li Xue-Hu;  Yi Yun-Peng;  Lu Xi-Hong;  Wang Liang
收藏  |  浏览/下载:21/0  |  提交时间:2018/05/31
A two-dimensional molecule with a large conjugation degree: synthesis, two-photon absorption and charge transport ability 期刊论文
JOURNAL OF MATERIALS CHEMISTRY C, 2017, 卷号: 5, 期号: 21, 页码: 5199-5206
作者:  Chen, Dugang;  Zhong, Cheng;  Zhao, Yan;  Nan, Lingyan;  Liu, Yunqi
收藏  |  浏览/下载:16/0  |  提交时间:2018/04/10
Synthesis and structure-activity relationship study of pyrazolo[3,4-d]pyrimidines as tyrosine kinase RET inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 11, 页码: 2544-2548
作者:  Wang, Chengyan;  Liu, Hongchun;  Song, Zilan;  Ji, Yinchun;  Xing, Li
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
嘧啶并吡啶酮骨架作为新型蛋白激酶小分子抑制剂的设计、合成及生物活性研究 学位论文
广州生物院: 中国科学院大学, 2017
作者:  余蕾
收藏  |  浏览/下载:439/0  |  提交时间:2018/12/25
Design, Synthesis and Anti-Proliferative Activities of 2,6-Substituted Thieno[3,2-d] pyrimidine Derivatives Containing ElectrophilicWarheads 期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 5
作者:  Zhang, Qiumeng;  Hu, Zonglong;  Shen, Qianqian;  Chen, Yi;  Lu, Wei
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
嘧啶衍生物类PI3K/mTOR双重抑制剂的3D-QSAR及分子对接研究 3D-QSAR and Surflex-dock study of pyrimidine scaffold compounds as dual PI3K/mTOR inhibitors 期刊论文
2017, 卷号: 47, 页码: 865-875
作者:  汪斌[1];  刘蒙蒙[1];  周朋朋[1];  林治华[1,2]
收藏  |  浏览/下载:3/0  |  提交时间:2019/11/30
Installation of biologically active pyrimidine moiety into pyridopyrimidine framework and evaluation of their antibacterial activities 期刊论文
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 2017, 卷号: 56, 页码: 120-126
作者:  Majumdar, Poulomi;  Pattnaik, Smaranika;  Dash, Debashrita;  Mohanta, Prajna Parimita;  Behera, Ajaya Kumar
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/02
Design, synthesis and biological evaluation of [1,2,4]triazolo[1,5-a]pyrimidines as potent lysine specific demethylase 1 (LSD1/KDM1A) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 125, 页码: 940-951
作者:  Wang, Shuai;  Zhao, Li-Jie;  Zheng, Yi-Chao;  Shen, Dan-Dan;  Miao, Er-Fei
收藏  |  浏览/下载:10/0  |  提交时间:2019/12/03
Design, Synthesis, and Biological Activity of Tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine Derivatives as Anti-Inflammatory Agents 期刊论文
MOLECULES, 2017, 卷号: 22
作者:  Zhang, Yuan;  Luo, Lu;  Han, Chao;  Lv, Handeng;  Chen, Di
收藏  |  浏览/下载:6/0  |  提交时间:2019/11/26


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