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Design, Synthesis, and Pharmacological Evaluation of 2-(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)-N-aryl Propanamides as Novel Smoothened (Smo) Antagonists 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 24, 页码: 11050-11068
作者:  Liu, Gang;  Xue, Ding;  Yang, Jun;  Wan, Juan;  Liu, Xiaohua
收藏  |  浏览/下载:54/0  |  提交时间:2019/01/08
Elucidating the druggable interface of protein-protein interactions using fragment docking and coevolutionary analysis 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2016, 卷号: 113, 期号: 50, 页码: E8051-E8058
作者:  Bai, Fang;  Morcos, Faruck;  Cheng, Ryan R.;  Jiang, Hualiang;  Onuchic, Jose N.
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Multivalent S-sialoside protein conjugates block influenza hemagglutinin and neuraminidase 期刊论文
CARBOHYDRATE RESEARCH, 2016, 卷号: 435, 页码: 68-75
作者:  Yang, Yang;  Liu, Hai-Peng;  Yu, Qun;  Yang, Mei-Bing;  Wang, De-Min
收藏  |  浏览/下载:40/0  |  提交时间:2017/03/13
Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 22, 页码: 10329-10334
作者:  Zhou, Pengfei;  Liu, Yan;  Zhou, Lu;  Zhu, Kongkai;  Feng, Kechang
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Rational design of multi-targeting ruthenium- and platinum-based anticancer complexes 期刊论文
SCIENCE CHINA-CHEMISTRY, 2016, 卷号: 59, 期号: 10, 页码: 1240-1249
作者:  Zheng, Wei;  Zhao, Yao;  Luo, Qun;  Zhang, Yang;  Wu, Kui
收藏  |  浏览/下载:73/0  |  提交时间:2017/01/17
Glucagon-Like Peptide-1 and Its Class B G Protein-Coupled Receptors: A Long March to Therapeutic Successes 期刊论文
PHARMACOLOGICAL REVIEWS, 2016, 卷号: 68, 期号: 4, 页码: 954-1013
作者:  de Graaf, Chris;  Donnelly, Dan;  Wootten, Denise;  Lau, Jesper;  Sexton, Patrick M.
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Synthesis and Anti-HIV-1 Activity Evaluation for Novel 3a,6a-Dihydro-1H-pyrrolo[3,4-c]pyrazole-4,6-dione Derivatives 期刊论文
MOLECULES, 2016, 卷号: 21, 期号: 9
作者:  Liu, Guan-Nan;  Luo, Rong-Hua;  Zhou, Yu;  Zhang, Xing-Jie;  Li, Jian
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Discovery and Structural Optimization of N5-Substituted 6,7-Dioxo-6,7-dihydropteridines as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 15, 页码: 7111-7124
作者:  Hao, Yongjia;  Wang, Xia;  Zhang, Tao;  Sun, Deheng;  Tong, Yi
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
A comparative study on the interactions of human copper chaperone Cox17 with anticancer organoruthenium(II) complexes and cisplatin by mass spectrometry 期刊论文
JOURNAL OF INORGANIC BIOCHEMISTRY, 2016, 卷号: 161, 页码: 99-106
作者:  Li, Lijie;  Guo, Wei;  Wu, Kui;  Wu, Xuelei;  Zhao, Linhong
收藏  |  浏览/下载:34/0  |  提交时间:2017/01/11
A Novel Bufalin Derivative Exhibited Stronger Apoptosis-Inducing Effect than Bufalin in A549 Lung Cancer Cells and Lower Acute Toxicity in Mice 期刊论文
PLOS ONE, 2016, 卷号: 11, 期号: 7
作者:  Liu, Miao;  Feng, Li-Xing;  Sun, Peng;  Liu, Wang;  Wu, Wan-Ying
收藏  |  浏览/下载:9/0  |  提交时间:2019/01/08


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