Progress in the Synthesis of Primary Anilines via C-H Bond Functionalization

doi:10.6023/cjoc201804004

	Progress in the Synthesis of Primary Anilines via C-H Bond Functionalization
	Xu, Linlin 1; Xu, Hui 3; Lin, Haixia 1; Dai, Huixiong2
刊名	CHINESE JOURNAL OF ORGANIC CHEMISTRY
	2018-08-25
卷号	38 期号:8 页码:1940-1948
关键词	amination C-H bond functionalization primary anilines transition-metal catalyzed
ISSN号	0253-2786
DOI	10.6023/cjoc201804004
文献子类	Review
英文摘要	Primary anilines are widely used in pharmaceutical, agrochemicals and material chemistry. In recent years, the green and efficient methods for constructing carbon-nitrogen (C-N) bonds to introduce primary amines has been one of the hottest topics in chemical synthesis. The direct C-H primary amination of aromatic compounds have received considerable attention due to its high efficiency and practicality. The recent progress in the C-H primary amination of aromatic compounds reactions is reviewed. Furthermore, the synthetic challenge and prospect in the future development for the synthesis of primary anilines through direct C-H amination are summarized.
资助项目	National Natural Science Foundation of China[21772211] ; Youth Innovation Promotion Association of Chinese Academy of Sciences[2014229]
WOS关键词	CROSS-COUPLING REACTIONS ; CARBON-HYDROGEN BONDS ; AROMATIC AMINATION ; ROOM-TEMPERATURE ; CUPRIC ACETATE ; STEP AMINATION ; PRIMARY AMINES ; COPPER ; ACTIVATION ; AMIDATION
WOS研究方向	Chemistry
语种	中文
CSCD记录号	CSCD:6321998
出版者	SCIENCE PRESS
WOS记录号	WOS:000450199700008
内容类型	期刊论文
源URL	[http://119.78.100.183/handle/2S10ELR8/279610]
专题	药物化学研究室
通讯作者	Lin, Haixia; Dai, Huixiong
作者单位	1.Shanghai Univ, Dept Chem, Innovat Drug Res Ctr, Shanghai 200444, Peoples R China; 2.Chinese Acad Sci, Dept Med Chem, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China; 3.Chinese Acad Sci, State Key Lab Organometall Chem, Shanghai Inst Organ Chem, Shanghai 200032, Peoples R China
推荐引用方式 GB/T 7714	Xu, Linlin,Xu, Hui,Lin, Haixia,et al. Progress in the Synthesis of Primary Anilines via C-H Bond Functionalization[J]. CHINESE JOURNAL OF ORGANIC CHEMISTRY,2018,38(8):1940-1948.
APA	Xu, Linlin,Xu, Hui,Lin, Haixia,&Dai, Huixiong.(2018).Progress in the Synthesis of Primary Anilines via C-H Bond Functionalization.CHINESE JOURNAL OF ORGANIC CHEMISTRY,38(8),1940-1948.
MLA	Xu, Linlin,et al."Progress in the Synthesis of Primary Anilines via C-H Bond Functionalization".CHINESE JOURNAL OF ORGANIC CHEMISTRY 38.8(2018):1940-1948.