Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization Process

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	Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization Process
	Shi L(石柳) ; Liu XQ(刘向前) ; Zhang H(张慧) ; Jiang YW(蒋咏文) ; Ma DW(马大为)
刊名	J. Org. Chem.
	2011
卷号	76 期号:10 页码:4200-4204
ISSN号	0022-3263
其他题名	经由一个多米诺缩合/S-芳基化/杂环化反应合成2-S-取代苯并噻唑
通讯作者	马大为
英文摘要	Condensation of carbon disulfide with thiols in the presence of K(2)CO(3) generates carbonotrithioate salts in situ, which undergo coupling with 2-iodoanilines and subsequent intramolecular condensation and elimination under assistance of CuBr to afford 2-thio-substituted benzothiazoles. Both aliphatic and aromatic thiols are compatible with this process, delivering the corresponding heterocycles with good diversity.
学科主题	有机化学
收录类别	SCI
原文出处	http://dx.doi.org/10.1021/jo200535e
语种	英语
WOS记录号	WOS:000290465700072
公开日期	2013-02-19
内容类型	期刊论文
源URL	[http://202.127.28.38/handle/331003/15667]
专题	上海有机化学研究所_生命有机化学国家重点实验室
推荐引用方式 GB/T 7714	Shi L,Liu XQ,Zhang H,et al. Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization Process[J]. J. Org. Chem.,2011,76(10):4200-4204.
APA	石柳,刘向前,张慧,蒋咏文,&马大为.(2011).Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization Process.J. Org. Chem.,76(10),4200-4204.
MLA	石柳,et al."Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization Process".J. Org. Chem. 76.10(2011):4200-4204.