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Design, synthesis and pharmacological evaluation of chalcone derivatives as acetylcholinesterase inhibitors
Liu, Hao-ran*; Liu, Xian-jun; Fan, Hao-qun; Tang, Jing-jing; Gao, Xiao-hui; Liu, Wu-kun
刊名Bioorganic and Medicinal Chemistry
2014
卷号22期号:21页码:6124-6133
关键词AD Alzheimer’s disease AChE acetylcholinesterases ACh acetylcholine BuChE butyrylcholinesterase PAS peripheral anionic sites Log P octanol/water partition CNS central nervous system BBB blood brain barrier Chalcone derivatives AChE inhibitors Log P Molecular docking
ISSN号0968-0896
DOI10.1016/j.bmc.2014.08.033
URL标识查看原文
WOS记录号WOS:000344471800041
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/5706251
专题湖南中医药大学
作者单位1.[Liu, Hao-ran
2.Liu, Wu-kun
3.Liu, Xian-jun
4.Fan, Hao-qun
5.Tang, Jing-jing] Hunan Univ, Coll Chem & Chem Engn, Changsha 410082, Hunan, Peoples R China.
推荐引用方式
GB/T 7714
Liu, Hao-ran*,Liu, Xian-jun,Fan, Hao-qun,et al. Design, synthesis and pharmacological evaluation of chalcone derivatives as acetylcholinesterase inhibitors[J]. Bioorganic and Medicinal Chemistry,2014,22(21):6124-6133.
APA Liu, Hao-ran*,Liu, Xian-jun,Fan, Hao-qun,Tang, Jing-jing,Gao, Xiao-hui,&Liu, Wu-kun.(2014).Design, synthesis and pharmacological evaluation of chalcone derivatives as acetylcholinesterase inhibitors.Bioorganic and Medicinal Chemistry,22(21),6124-6133.
MLA Liu, Hao-ran*,et al."Design, synthesis and pharmacological evaluation of chalcone derivatives as acetylcholinesterase inhibitors".Bioorganic and Medicinal Chemistry 22.21(2014):6124-6133.
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