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Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site
Qinhuai Lai; Yuxi Wang; Ruixue Wang; Weirong Lai; Liangze Tang; Yiran Tao; Yu Liu; Ruirui Zhang; Luyi Huang; Haotian Xiang
刊名European Journal of Medicinal Chemistry
2018
关键词Tubulin inhibitor Colchicine binding site Combretastatin A-4 Pyrazole analogue Anti-tumour Co-crystal structure
ISSN号0223-5234
URL标识查看原文
内容类型期刊论文
URI标识http://www.corc.org.cn/handle/1471x/1870634
专题四川大学
作者单位1.b State Key Laboratory of Biotherapy and Cancer Center/Collaborative Innovation Center for Biotherapy, West China Hospital, Sichuan University, Chengdu, PR China a Research Center for Public Health and Preventive Medicine/Research Center for Occupational Respiratory Diseases, West China School of Public Health and Healthy Food Evaluation Research Center /No
2.Ophthalmic Laboratories & Department of Ophthalmology, Translational Neuroscience Center, West China Hospital, Sichuan University, Chengdu, PR China
3.West China Teaching Hospital, Sichuan University, Chengdu, PR China
4.Guangdong Zhongsheng Pharmaceutical Co., Ltd., China
推荐引用方式
GB/T 7714
Qinhuai Lai,Yuxi Wang,Ruixue Wang,et al. Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site[J]. European Journal of Medicinal Chemistry,2018.
APA Qinhuai Lai.,Yuxi Wang.,Ruixue Wang.,Weirong Lai.,Liangze Tang.,...&Jinliang Yang.(2018).Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site.European Journal of Medicinal Chemistry.
MLA Qinhuai Lai,et al."Design, synthesis and biological evaluation of a novel tubulin inhibitor 7a3 targeting the colchicine binding site".European Journal of Medicinal Chemistry (2018).
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