Efficient synthesis of 5-fluroalkylated 1H-1,2,3-Triazoles and application of the bromodifloromethylated triazole toprepare new gem-difluorinated triazole compounds.

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	Efficient synthesis of 5-fluroalkylated 1H-1,2,3-Triazoles and application of the bromodifloromethylated triazole toprepare new gem-difluorinated triazole compounds.
	Peng WM(彭卫民) ; Zhu SZ(朱仕正)
刊名	Synlett
	2003
期号	2 页码:187-190
ISSN号	0936-5214
其他题名	高效合成5-氟烷基1H-1,2,3三氮唑和运用溴二氟甲基取代的三氮唑制备一些新的二氟亚甲基化的三氮唑化合物
通讯作者	朱仕正
英文摘要	A series of 5-fluoroalkylated 1H-1,2,3-triazoles was prepared in good yield by the regiospecific 1,3-dipolar cycloaddition reaction of the (Z) ethyl 3-fluoroalkyl-3-pyrrolidino-acrylates with aryl or benzyl azides. In the cases of benzyl azides, addition of Na^2CO^3 was crucial for a high yield of the triazoles. The tetrakis(dimethylamino)ethylene (TDAE) promoted reaction of the bromo-difluoromethylated 1H-1,2,3-triazole with aldehyde afforded a new class of novel gem-difluorinated triazole compounds.
学科主题	有机氟化学
收录类别	SCI
原文出处	http://dx.doi.org/10.1055/s-2003-36784
语种	英语
公开日期	2013-01-18
内容类型	期刊论文
源URL	[http://202.127.28.38/handle/331003/14292]
专题	上海有机化学研究所_中科院有机氟化学重点实验室
推荐引用方式 GB/T 7714	Peng WM,Zhu SZ. Efficient synthesis of 5-fluroalkylated 1H-1,2,3-Triazoles and application of the bromodifloromethylated triazole toprepare new gem-difluorinated triazole compounds.[J]. Synlett,2003(2):187-190.
APA	彭卫民,&朱仕正.(2003).Efficient synthesis of 5-fluroalkylated 1H-1,2,3-Triazoles and application of the bromodifloromethylated triazole toprepare new gem-difluorinated triazole compounds..Synlett(2),187-190.
MLA	彭卫民,et al."Efficient synthesis of 5-fluroalkylated 1H-1,2,3-Triazoles and application of the bromodifloromethylated triazole toprepare new gem-difluorinated triazole compounds.".Synlett .2(2003):187-190.