A Facile Approach to Optically Active Hydroquinoline-2-carboxylates by a One-Pot Asymmetric Michael/Transamination/Cyclization Process

	A Facile Approach to Optically Active Hydroquinoline-2-carboxylates by a One-Pot Asymmetric Michael/Transamination/Cyclization Process
	Rong, Chao 1; Pan, Hongjie 1; Liu, Mao 1; Tian, Hua 1; Shi, Yian 1,2
刊名	CHEMISTRY-A EUROPEAN JOURNAL
	2016-02-24
卷号	22 期号:9 页码:2887-2891
关键词	cyclization Michael addition organocatalysis transamination
英文摘要	An efficient one-pot synthesis of optically active hydroquinoline-2-carboxylates from 1,3-cyclohexanediones, ,-unsaturated -keto ester, and benzylamine in the presence of a chiral base catalyst and 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU) with good diastereoselectivity and high enantioselectivity is described. The reaction proceeds by a sequential asymmetric Michael/transamination/cyclization process.
收录类别	SCI
语种	英语
内容类型	期刊论文
源URL	[http://ir.iccas.ac.cn/handle/121111/35821]
专题	化学研究所_分子识别与功能实验室
作者单位	1.Chinese Acad Sci, Inst Chem, Beijing Natl Lab Mol Sci, CAS Key Lab Mol Recognit & Funct, Beijing 100190, Peoples R China 2.Colorado State Univ, Dept Chem, Ft Collins, CO 80523 USA
推荐引用方式 GB/T 7714	Rong, Chao,Pan, Hongjie,Liu, Mao,et al. A Facile Approach to Optically Active Hydroquinoline-2-carboxylates by a One-Pot Asymmetric Michael/Transamination/Cyclization Process[J]. CHEMISTRY-A EUROPEAN JOURNAL,2016,22(9):2887-2891.
APA	Rong, Chao,Pan, Hongjie,Liu, Mao,Tian, Hua,&Shi, Yian.(2016).A Facile Approach to Optically Active Hydroquinoline-2-carboxylates by a One-Pot Asymmetric Michael/Transamination/Cyclization Process.CHEMISTRY-A EUROPEAN JOURNAL,22(9),2887-2891.
MLA	Rong, Chao,et al."A Facile Approach to Optically Active Hydroquinoline-2-carboxylates by a One-Pot Asymmetric Michael/Transamination/Cyclization Process".CHEMISTRY-A EUROPEAN JOURNAL 22.9(2016):2887-2891.